Abulkhair HS - Search Results

1

Arylthiazole antibiotics targeting intracellular methicillin-resistant Staphylococcus aureus (MRSA) that interfere with bacterial cell wall synthesis.

Eid I, Elsebaei MM, Mohammad H, Hagras M, Peters CE, Hegazy YA, Cooper B, Pogliano J, Pogliano K, Abulkhair HS, Seleem MN, Mayhoub AS. Eid I, et al. Among authors: abulkhair hs. Eur J Med Chem. 2017 Oct 20;139:665-673. doi: 10.1016/j.ejmech.2017.08.039. Epub 2017 Aug 18. Eur J Med Chem. 2017. PMID: 28846967 Free PMC article.

2

Synthesis and antibacterial evaluation of a novel library of 2-(thiazol-5-yl)-1,3,4-oxadiazole derivatives against methicillin-resistant Staphylococcus aureus (MRSA).

Hannoun MH, Hagras M, Kotb A, El-Attar AMM, Abulkhair HS. Hannoun MH, et al. Among authors: abulkhair hs. Bioorg Chem. 2020 Jan;94:103364. doi: 10.1016/j.bioorg.2019.103364. Epub 2019 Oct 18. Bioorg Chem. 2020. PMID: 31668461

3

From triazolophthalazines to triazoloquinazolines: A bioisosterism-guided approach toward the identification of novel PCAF inhibitors with potential anticancer activity.

El-Shershaby MH, Ghiaty A, Bayoumi AH, Al-Karmalawy AA, Husseiny EM, El-Zoghbi MS, Abulkhair HS. El-Shershaby MH, et al. Among authors: abulkhair hs. Bioorg Med Chem. 2021 Jul 15;42:116266. doi: 10.1016/j.bmc.2021.116266. Epub 2021 Jun 5. Bioorg Med Chem. 2021. PMID: 34126285

4

Rational design, synthesis, pharmacophore modeling, and docking studies for identification of novel potent DNA-PK inhibitors.

Ihmaid S, Ahmed HEA, Al-Sheikh Ali A, Sherif YE, Tarazi HM, Riyadh SM, Zayed MF, Abulkhair HS, Rateb HS. Ihmaid S, et al. Among authors: abulkhair hs. Bioorg Chem. 2017 Jun;72:234-247. doi: 10.1016/j.bioorg.2017.04.014. Epub 2017 May 2. Bioorg Chem. 2017. PMID: 28482264

5

Design, synthesis, in silico ADMET profile and GABA-A docking of novel phthalazines as potent anticonvulsants.

El-Helby AA, Ayyad RRA, Zayed MF, Abulkhair HS, Elkady H, El-Adl K. El-Helby AA, et al. Among authors: abulkhair hs. Arch Pharm (Weinheim). 2019 May;352(5):e1800387. doi: 10.1002/ardp.201800387. Epub 2019 Apr 15. Arch Pharm (Weinheim). 2019. PMID: 30989729

6

Design, synthesis, molecular docking, and anticancer activity of benzoxazole derivatives as VEGFR-2 inhibitors.

El-Helby AA, Sakr H, Eissa IH, Abulkhair H, Al-Karmalawy AA, El-Adl K. El-Helby AA, et al. Arch Pharm (Weinheim). 2019 Oct;352(10):e1900113. doi: 10.1002/ardp.201900113. Epub 2019 Aug 25. Arch Pharm (Weinheim). 2019. PMID: 31448458

7

The rational design, synthesis, and antimicrobial investigation of 2-Amino-4-Methylthiazole analogues inhibitors of GlcN-6-P synthase.

Omar AM, Ihmaid S, Habib EE, Althagfan SS, Ahmed S, Abulkhair HS, Ahmed HEA. Omar AM, et al. Among authors: abulkhair hs. Bioorg Chem. 2020 Jun;99:103781. doi: 10.1016/j.bioorg.2020.103781. Epub 2020 Mar 21. Bioorg Chem. 2020. PMID: 32222620

8

Design, synthesis, and antitumor activity of novel compounds based on 1,2,4-triazolophthalazine scaffold: Apoptosis-inductive and PCAF-inhibitory effects.

Turky A, Bayoumi AH, Ghiaty A, El-Azab AS, A-M Abdel-Aziz A, Abulkhair HS. Turky A, et al. Among authors: abulkhair hs. Bioorg Chem. 2020 Aug;101:104019. doi: 10.1016/j.bioorg.2020.104019. Epub 2020 Jun 17. Bioorg Chem. 2020. PMID: 32615465

9

Unravelling the anticancer potency of 1,2,4-triazole-N-arylamide hybrids through inhibition of STAT3: synthesis and in silico mechanistic studies.

Turky A, Bayoumi AH, Sherbiny FF, El-Adl K, Abulkhair HS. Turky A, et al. Among authors: abulkhair hs. Mol Divers. 2021 Feb;25(1):403-420. doi: 10.1007/s11030-020-10131-0. Epub 2020 Aug 23. Mol Divers. 2021. PMID: 32830299

10

Novel 1,2,4-triazole derivatives: Design, synthesis, anticancer evaluation, molecular docking, and pharmacokinetic profiling studies.

Turky A, Sherbiny FF, Bayoumi AH, Ahmed HEA, Abulkhair HS. Turky A, et al. Among authors: abulkhair hs. Arch Pharm (Weinheim). 2020 Dec;353(12):e2000170. doi: 10.1002/ardp.202000170. Epub 2020 Sep 6. Arch Pharm (Weinheim). 2020. PMID: 32893368

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