Gao P - Search Results

1

1-Hydroxypyrido[2,3-d]pyrimidin-2(1H)-ones as novel selective HIV integrase inhibitors obtained via privileged substructure-based compound libraries.

Gao P, Zhang L, Sun L, Huang T, Tan J, Zhang J, Zhou Z, Zhao T, Menéndez-Arias L, Pannecouque C, Clercq E, Zhan P, Liu X. Gao P, et al. Bioorg Med Chem. 2017 Oct 15;25(20):5779-5789. doi: 10.1016/j.bmc.2017.09.006. Epub 2017 Sep 8. Bioorg Med Chem. 2017. PMID: 28951095

2

Design, Synthesis, and Mechanism Study of Benzenesulfonamide-Containing Phenylalanine Derivatives as Novel HIV-1 Capsid Inhibitors with Improved Antiviral Activities.

Sun L, Dick A, Meuser ME, Huang T, Zalloum WA, Chen CH, Cherukupalli S, Xu S, Ding X, Gao P, Kang D, De Clercq E, Pannecouque C, Cocklin S, Lee KH, Liu X, Zhan P. Sun L, et al. Among authors: gao p. J Med Chem. 2020 May 14;63(9):4790-4810. doi: 10.1021/acs.jmedchem.0c00015. Epub 2020 Apr 29. J Med Chem. 2020. PMID: 32298111 Free PMC article.

3

Discovery of potential dual-target prodrugs of HIV-1 reverse transcriptase and nucleocapsid protein 7.

Sun S, Huang B, Li Z, Wang Z, Sun L, Gao P, Kang D, Chen CH, Lee KH, Daelemans D, De Clercq E, Pannecouque C, Zhan P, Liu X. Sun S, et al. Among authors: gao p. Bioorg Med Chem Lett. 2020 Aug 15;30(16):127287. doi: 10.1016/j.bmcl.2020.127287. Epub 2020 May 26. Bioorg Med Chem Lett. 2020. PMID: 32631509

4

Novel indolylarylsulfone derivatives as covalent HIV-1 reverse transcriptase inhibitors specifically targeting the drug-resistant mutant Y181C.

Gao P, Song S, Frutos-Beltrán E, Li W, Sun B, Kang D, Zou J, Zhang J, Pannecouque C, De Clercq E, Menéndez-Arias L, Zhan P, Liu X. Gao P, et al. Bioorg Med Chem. 2021 Jan 15;30:115927. doi: 10.1016/j.bmc.2020.115927. Epub 2020 Dec 10. Bioorg Med Chem. 2021. PMID: 33352387 Free article.

5

Design, synthesis and anti-HIV evaluation of novel 5-substituted diarylpyrimidine derivatives as potent HIV-1 NNRTIs.

Gao P, Song S, Wang Z, Sun L, Zhang J, Pannecouque C, De Clercq E, Zhan P, Liu X. Gao P, et al. Bioorg Med Chem. 2021 Jun 15;40:116195. doi: 10.1016/j.bmc.2021.116195. Epub 2021 May 5. Bioorg Med Chem. 2021. PMID: 33979774

6

Structure-Based Design and Discovery of Pyridyl-Bearing Fused Bicyclic HIV-1 Inhibitors: Synthesis, Biological Characterization, and Molecular Modeling Studies.

Huang B, Ginex T, Luque FJ, Jiang X, Gao P, Zhang J, Kang D, Daelemans D, De Clercq E, Pannecouque C, Zhan P, Liu X. Huang B, et al. Among authors: gao p. J Med Chem. 2021 Sep 23;64(18):13604-13621. doi: 10.1021/acs.jmedchem.1c00987. Epub 2021 Sep 9. J Med Chem. 2021. PMID: 34496571

7

Indolylarylsulfones bearing phenylboronic acid and phenylboronate ester functionalities as potent HIV‑1 non-nucleoside reverse transcriptase inhibitors.

Xu S, Song S, Sun L, Gao P, Gao S, Ma Y, Kang D, Cheng Y, Zhang X, Cherukupalli S, De Clercq E, Pannecouque C, Liu X, Zhan P. Xu S, et al. Among authors: gao s, gao p. Bioorg Med Chem. 2022 Jan 1;53:116531. doi: 10.1016/j.bmc.2021.116531. Epub 2021 Dec 3. Bioorg Med Chem. 2022. PMID: 34890994

8

Chemical space exploration around indolylarylsulfone scaffold led to a novel class of highly active HIV-1 NNRTIs with spiro structural features.

Gao S, Cheng Y, Song S, Song L, Zhao F, Xu S, Kang D, Sun L, Gao P, De Clercq E, Pannecouque C, Liu X, Zhan P. Gao S, et al. Among authors: gao p. Eur J Med Chem. 2022 Aug 5;238:114471. doi: 10.1016/j.ejmech.2022.114471. Epub 2022 May 20. Eur J Med Chem. 2022. PMID: 35640327

9

Identification of spirocyclic or phosphate substituted quinolizine derivatives as novel HIV-1 integrase inhibitors: a patent evaluation of WO2016094197A1, WO2016094198A1 and WO2016154527A1.

Cheng X, Gao P, Sun L, Tian Y, Zhan P, Liu X. Cheng X, et al. Among authors: gao p. Expert Opin Ther Pat. 2017 Nov;27(11):1277-1286. doi: 10.1080/13543776.2017.1360283. Epub 2017 Aug 2. Expert Opin Ther Pat. 2017. PMID: 28749251 Review.

10

The discovery of novel diarylpyri(mi)dine derivatives with high level activity against a wide variety of HIV-1 strains as well as against HIV-2.

Lu X, Yang J, Kang D, Gao P, Daelemans D, De Clercq E, Pannecouque C, Zhan P, Liu X. Lu X, et al. Among authors: gao p. Bioorg Med Chem. 2018 May 1;26(8):2051-2060. doi: 10.1016/j.bmc.2018.03.003. Epub 2018 Mar 3. Bioorg Med Chem. 2018. PMID: 29559197

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