Krasavin M - Search Results

1

Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII.

Kalinin S, Kopylov S, Tuccinardi T, Sapegin A, Dar'in D, Angeli A, Supuran CT, Krasavin M. Kalinin S, et al. Among authors: krasavin m. ACS Med Chem Lett. 2017 Sep 15;8(10):1105-1109. doi: 10.1021/acsmedchemlett.7b00300. eCollection 2017 Oct 12. ACS Med Chem Lett. 2017. PMID: 29057059 Free PMC article.

2

Probing the 'bipolar' nature of the carbonic anhydrase active site: aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms.

Krasavin M, Korsakov M, Dorogov M, Tuccinardi T, Dedeoglu N, Supuran CT. Krasavin M, et al. Eur J Med Chem. 2015 Aug 28;101:334-47. doi: 10.1016/j.ejmech.2015.06.022. Epub 2015 Jun 25. Eur J Med Chem. 2015. PMID: 26160114

3

New Heterocyclic Product Space for the Castagnoli-Cushman Three-Component Reaction.

Dar'in D, Bakulina O, Chizhova M, Krasavin M. Dar'in D, et al. Among authors: krasavin m. Org Lett. 2015 Aug 7;17(15):3930-3. doi: 10.1021/acs.orglett.5b02014. Epub 2015 Jul 30. Org Lett. 2015. PMID: 26226189

4

Discovery of Strecker-type α-aminonitriles as a new class of human carbonic anhydrase inhibitors using differential scanning fluorimetry.

Krasavin M, Stavniichuk R, Zozulya S, Borysko P, Vullo D, Supuran CT. Krasavin M, et al. J Enzyme Inhib Med Chem. 2016 Dec;31(6):1707-11. doi: 10.3109/14756366.2016.1156676. Epub 2016 Mar 16. J Enzyme Inhib Med Chem. 2016. PMID: 26983069 Free article.

5

Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases.

Supuran CT, Kalinin S, Tanç M, Sarnpitak P, Mujumdar P, Poulsen SA, Krasavin M. Supuran CT, et al. Among authors: krasavin m. J Enzyme Inhib Med Chem. 2016;31(sup1):197-202. doi: 10.1080/14756366.2016.1178248. Epub 2016 May 10. J Enzyme Inhib Med Chem. 2016. PMID: 27160030 Free article.

6

Multicomponent chemistry in the synthesis of carbonic anhydrase inhibitors.

Kalinin S, Supuran CT, Krasavin M. Kalinin S, et al. Among authors: krasavin m. J Enzyme Inhib Med Chem. 2016;31(sup4):185-199. doi: 10.1080/14756366.2016.1220944. Epub 2016 Oct 26. J Enzyme Inhib Med Chem. 2016. PMID: 27784162 Free article. Review.

7

The Chan-Evans-Lam N-Arylation of 2-Imidazolines.

Dar'in D, Krasavin M. Dar'in D, et al. Among authors: krasavin m. J Org Chem. 2016 Dec 16;81(24):12514-12519. doi: 10.1021/acs.joc.6b02404. Epub 2016 Nov 30. J Org Chem. 2016. PMID: 27978721

8

Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds.

Krasavin M, Korsakov M, Zvonaryova Z, Semyonychev E, Tuccinardi T, Kalinin S, Tanç M, Supuran CT. Krasavin M, et al. Bioorg Med Chem. 2017 Mar 15;25(6):1914-1925. doi: 10.1016/j.bmc.2017.02.018. Epub 2017 Feb 13. Bioorg Med Chem. 2017. PMID: 28237553

9

Structurally diverse arene-fused ten-membered lactams accessed via hydrolytic imidazoline ring expansion.

Sapegin A, Osipyan A, Krasavin M. Sapegin A, et al. Among authors: krasavin m. Org Biomol Chem. 2017 Apr 5;15(14):2906-2909. doi: 10.1039/c7ob00535k. Org Biomol Chem. 2017. PMID: 28321443

10

Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases.

Krasavin M, Korsakov M, Ronzhina O, Tuccinardi T, Kalinin S, Tanç M, Supuran CT. Krasavin M, et al. J Enzyme Inhib Med Chem. 2017 Dec;32(1):920-934. doi: 10.1080/14756366.2017.1344236. J Enzyme Inhib Med Chem. 2017. PMID: 28718328 Free PMC article.

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