Zhu Y - Search Results

1

Structure-Activity Relationship Studies with Tetrahydroquinoline Analogs as EPAC Inhibitors.

Sonawane YA, Zhu Y, Garrison JC, Ezell EL, Zahid M, Cheng X, Natarajan A. Sonawane YA, et al. Among authors: zhu y. ACS Med Chem Lett. 2017 Oct 2;8(11):1183-1187. doi: 10.1021/acsmedchemlett.7b00358. eCollection 2017 Nov 9. ACS Med Chem Lett. 2017. PMID: 29375750 Free PMC article.

2

Structure-Activity Relationship Studies of Substituted 2-(Isoxazol-3-yl)-2-oxo-N'-phenyl-acetohydrazonoyl Cyanide Analogues: Identification of Potent Exchange Proteins Directly Activated by cAMP (EPAC) Antagonists.

Ye N, Zhu Y, Chen H, Liu Z, Mei FC, Wild C, Chen H, Cheng X, Zhou J. Ye N, et al. Among authors: zhu y. J Med Chem. 2015 Aug 13;58(15):6033-47. doi: 10.1021/acs.jmedchem.5b00635. Epub 2015 Jul 16. J Med Chem. 2015. PMID: 26151319 Free PMC article.

3

Functionalized N,N-Diphenylamines as Potent and Selective EPAC2 Inhibitors.

Wild CT, Zhu Y, Na Y, Mei F, Ynalvez MA, Chen H, Cheng X, Zhou J. Wild CT, et al. Among authors: zhu y. ACS Med Chem Lett. 2016 Mar 28;7(5):460-4. doi: 10.1021/acsmedchemlett.5b00477. eCollection 2016 May 12. ACS Med Chem Lett. 2016. PMID: 27190593 Free PMC article.

4

Structure-activity relationships of 2-substituted phenyl-N-phenyl-2-oxoacetohydrazonoyl cyanides as novel antagonists of exchange proteins directly activated by cAMP (EPACs).

Liu Z, Zhu Y, Chen H, Wang P, Mei FC, Ye N, Cheng X, Zhou J. Liu Z, et al. Among authors: zhu y. Bioorg Med Chem Lett. 2017 Dec 1;27(23):5163-5166. doi: 10.1016/j.bmcl.2017.10.056. Epub 2017 Oct 25. Bioorg Med Chem Lett. 2017. PMID: 29100797 Free PMC article.

5

Identification of novel 2-(benzo[d]isoxazol-3-yl)-2-oxo-N-phenylacetohydrazonoyl cyanide analoguesas potent EPAC antagonists.

Ye N, Zhu Y, Liu Z, Mei FC, Chen H, Wang P, Cheng X, Zhou J. Ye N, et al. Among authors: zhu y. Eur J Med Chem. 2017 Jul 7;134:62-71. doi: 10.1016/j.ejmech.2017.04.001. Epub 2017 Apr 4. Eur J Med Chem. 2017. PMID: 28399451 Free PMC article.

6

A cell-based, quantitative and isoform-specific assay for exchange proteins directly activated by cAMP.

Zhu Y, Mei F, Luo P, Cheng X. Zhu Y, et al. Sci Rep. 2017 Jul 24;7(1):6200. doi: 10.1038/s41598-017-06432-4. Sci Rep. 2017. PMID: 28740152 Free PMC article.

7

Biochemical and pharmacological characterizations of ESI-09 based EPAC inhibitors: defining the ESI-09 "therapeutic window".

Zhu Y, Chen H, Boulton S, Mei F, Ye N, Melacini G, Zhou J, Cheng X. Zhu Y, et al. Sci Rep. 2015 Mar 20;5:9344. doi: 10.1038/srep09344. Sci Rep. 2015. PMID: 25791905 Free PMC article.

8

Critical role for Epac1 in inflammatory pain controlled by GRK2-mediated phosphorylation of Epac1.

Singhmar P, Huo X, Eijkelkamp N, Berciano SR, Baameur F, Mei FC, Zhu Y, Cheng X, Hawke D, Mayor F Jr, Murga C, Heijnen CJ, Kavelaars A. Singhmar P, et al. Among authors: zhu y. Proc Natl Acad Sci U S A. 2016 Mar 15;113(11):3036-41. doi: 10.1073/pnas.1516036113. Epub 2016 Feb 29. Proc Natl Acad Sci U S A. 2016. PMID: 26929333 Free PMC article.

9

Rp-cAMPS Prodrugs Reveal the cAMP Dependence of First-Phase Glucose-Stimulated Insulin Secretion.

Schwede F, Chepurny OG, Kaufholz M, Bertinetti D, Leech CA, Cabrera O, Zhu Y, Mei F, Cheng X, Manning Fox JE, MacDonald PE, Genieser HG, Herberg FW, Holz GG. Schwede F, et al. Among authors: zhu y. Mol Endocrinol. 2015 Jul;29(7):988-1005. doi: 10.1210/me.2014-1330. Epub 2015 Jun 10. Mol Endocrinol. 2015. PMID: 26061564 Free PMC article.

10

Pyrazolopyrimidines as Potent Stimulators for Transient Receptor Potential Canonical 3/6/7 Channels.

Qu C, Ding M, Zhu Y, Lu Y, Du J, Miller M, Tian J, Zhu J, Xu J, Wen M, Er-Bu A, Wang J, Xiao Y, Wu M, McManus OB, Li M, Wu J, Luo HR, Cao Z, Shen B, Wang H, Zhu MX, Hong X. Qu C, et al. Among authors: zhu y, zhu j, zhu mx. J Med Chem. 2017 Jun 8;60(11):4680-4692. doi: 10.1021/acs.jmedchem.7b00304. Epub 2017 Apr 28. J Med Chem. 2017. PMID: 28395140 Free PMC article.

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