Le Borgne M - Search Results

1

2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 2. Structure-Based Optimization and Investigation of Effects Specific to the Allosteric Mode of Action.

Bestgen B, Kufareva I, Seetoh W, Abell C, Hartmann RW, Abagyan R, Le Borgne M, Filhol O, Cochet C, Lomberget T, Engel M. Bestgen B, et al. Among authors: le borgne m. J Med Chem. 2019 Feb 28;62(4):1817-1836. doi: 10.1021/acs.jmedchem.8b01765. Epub 2019 Feb 13. J Med Chem. 2019. PMID: 30689946 Free PMC article.

2

Synthesis and in vitro evaluation of 3-(1-azolylmethyl)-1H-indoles and 3-(1-azolyl-1-phenylmethyl)-1H-indoles as inhibitors of P450 arom.

Le Borgne M, Marchand P, Duflos M, Delevoye-Seiller B, Piessard-Robert S, Le Baut G, Hartmann RW, Palzer M. Le Borgne M, et al. Among authors: le baut g. Arch Pharm (Weinheim). 1997 May;330(5):141-5. doi: 10.1002/ardp.19973300506. Arch Pharm (Weinheim). 1997. PMID: 9237426

3

New selective nonsteroidal aromatase inhibitors: synthesis and inhibitory activity of 2,3 or 5-(alpha-azolylbenzyl)-1H-indoles.

Le Borgne M, Marchand P, Delevoye-Seiller B, Robert JM, Le Baut G, Hartmann RW, Palzer M. Le Borgne M, et al. Among authors: le baut g. Bioorg Med Chem Lett. 1999 Feb 8;9(3):333-6. doi: 10.1016/s0960-894x(98)00737-9. Bioorg Med Chem Lett. 1999. PMID: 10091679

4

[Synthesis and biological evaluation of indole derivatives acting as anti-inflammatory or antitumoral drugs].

Le Borgne M, Duflos M, Le Baut G, Nicholls PJ, Hartmann RW. Le Borgne M, et al. Among authors: le baut g. Ann Pharm Fr. 2000 Oct;58(5):316-20. Ann Pharm Fr. 2000. PMID: 11060408 French.

5

Preparation and pharmacological profile of 7-(alpha-azolylbenzyl)-1H-indoles and indolines as new aromatase inhibitors.

Marchand P, Le Borgne M, Palzer M, Le Baut G, Hartmann RW. Marchand P, et al. Among authors: le baut g, le borgne m. Bioorg Med Chem Lett. 2003 May 5;13(9):1553-5. doi: 10.1016/s0960-894x(03)00182-3. Bioorg Med Chem Lett. 2003. PMID: 12699753

6

2- and 3-[(aryl)(azolyl)methyl]indoles as potential non-steroidal aromatase inhibitors.

Lézé MP, Le Borgne M, Marchand P, Loquet D, Kogler M, Le Baut G, Palusczak A, Hartmann RW. Lézé MP, et al. Among authors: le baut g, le borgne m. J Enzyme Inhib Med Chem. 2004 Dec;19(6):549-57. doi: 10.1080/14756360400004631. J Enzyme Inhib Med Chem. 2004. PMID: 15662958 Free article.

7

Synthesis and biological evaluation of 5-[(aryl)(1H-imidazol-1-yl)methyl]-1H-indoles: potent and selective aromatase inhibitors.

Lézé MP, Le Borgne M, Pinson P, Palusczak A, Duflos M, Le Baut G, Hartmann RW. Lézé MP, et al. Among authors: le baut g, le borgne m. Bioorg Med Chem Lett. 2006 Mar 1;16(5):1134-7. doi: 10.1016/j.bmcl.2005.11.099. Epub 2005 Dec 27. Bioorg Med Chem Lett. 2006. PMID: 16380254

8

Three-dimensional model of cytochrome P450 human aromatase.

Loge C, Le Borgne M, Marchand P, Robert JM, Le Baut G, Palzer M, Hartmann RW. Loge C, et al. Among authors: le baut g, le borgne m. J Enzyme Inhib Med Chem. 2005 Dec;20(6):581-5. doi: 10.1080/14756360500220574. J Enzyme Inhib Med Chem. 2005. PMID: 16408794 Free article.

9

Synthesis and biological evaluation of 3-(azolylmethyl)-1H-indoles and 3-(alpha-azolylbenzyl)-1H-indoles as selective aromatase inhibitors.

Le Borgne M, Marchand P, Nourrisson MR, Loquet D, Palzer M, Le Baut G, Hartmann RW. Le Borgne M, et al. Among authors: le baut g. J Enzyme Inhib Med Chem. 2007 Oct;22(5):667-76. doi: 10.1080/14756360701652658. J Enzyme Inhib Med Chem. 2007. PMID: 18035835 Free article.

10

Synthesis of 6- or 4-functionalized indoles via a reductive cyclization approach and evaluation as aromatase inhibitors.

Lézé MP, Palusczak A, Hartmann RW, Le Borgne M. Lézé MP, et al. Among authors: le borgne m. Bioorg Med Chem Lett. 2008 Aug 15;18(16):4713-5. doi: 10.1016/j.bmcl.2008.06.094. Epub 2008 Jul 3. Bioorg Med Chem Lett. 2008. PMID: 18640836

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