Gao P - Search Results

1

Exploiting the Tolerant Region I of the Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI) Binding Pocket: Discovery of Potent Diarylpyrimidine-Typed HIV-1 NNRTIs against Wild-Type and E138K Mutant Virus with Significantly Improved Water Solubility and Favorable Safety Profiles.

Huang B, Chen W, Zhao T, Li Z, Jiang X, Ginex T, Vílchez D, Luque FJ, Kang D, Gao P, Zhang J, Tian Y, Daelemans D, De Clercq E, Pannecouque C, Zhan P, Liu X. Huang B, et al. Among authors: gao p. J Med Chem. 2019 Feb 28;62(4):2083-2098. doi: 10.1021/acs.jmedchem.8b01729. Epub 2019 Feb 20. J Med Chem. 2019. PMID: 30721060

2

Substituted indoles as HIV-1 non-nucleoside reverse transcriptase inhibitors: a patent evaluation (WO2015044928).

Li X, Gao P, Zhan P, Liu X. Li X, et al. Among authors: gao p. Expert Opin Ther Pat. 2016 May;26(5):629-35. doi: 10.1517/13543776.2016.1135902. Epub 2016 Feb 16. Expert Opin Ther Pat. 2016. PMID: 26742549

3

Arylazolyl(azinyl)thioacetanilides: Part 19: Discovery of Novel Substituted Imidazo[4,5-b]pyridin-2-ylthioacetanilides as Potent HIV NNRTIs Via a Structure-based Bioisosterism Approach.

Li X, Huang B, Zhou Z, Gao P, Pannecouque C, Daelemans D, De Clercq E, Zhan P, Liu X. Li X, et al. Among authors: gao p. Chem Biol Drug Des. 2016 Aug;88(2):241-53. doi: 10.1111/cbdd.12751. Epub 2016 Mar 24. Chem Biol Drug Des. 2016. PMID: 26914186

4

Pyrazolo[1,5-a]pyrimidine-based macrocycles as novel HIV-1 inhibitors: a patent evaluation of WO2015123182.

Sun L, Gao P, Zhan P, Liu X. Sun L, et al. Among authors: gao p. Expert Opin Ther Pat. 2016 Sep;26(9):979-86. doi: 10.1080/13543776.2016.1210127. Epub 2016 Jul 19. Expert Opin Ther Pat. 2016. PMID: 27398994

5

Discovery of novel anti-HIV agents via Cu(I)-catalyzed azide-alkyne cycloaddition (CuAAC) click chemistry-based approach.

Gao P, Sun L, Zhou J, Li X, Zhan P, Liu X. Gao P, et al. Expert Opin Drug Discov. 2016 Sep;11(9):857-71. doi: 10.1080/17460441.2016.1210125. Epub 2016 Jul 21. Expert Opin Drug Discov. 2016. PMID: 27400283 Review.

6

Discovery of novel piperidine-substituted indolylarylsulfones as potent HIV NNRTIs via structure-guided scaffold morphing and fragment rearrangement.

Li X, Gao P, Huang B, Zhou Z, Yu Z, Yuan Z, Liu H, Pannecouque C, Daelemans D, De Clercq E, Zhan P, Liu X. Li X, et al. Among authors: gao p. Eur J Med Chem. 2017 Jan 27;126:190-201. doi: 10.1016/j.ejmech.2016.10.009. Epub 2016 Oct 5. Eur J Med Chem. 2017. PMID: 27750153

7

Update on Recent Developments in Small Molecular HIV-1 RNase H Inhibitors (2013-2016): Opportunities and Challenges.

Wang X, Gao P, Menendez-Arias L, Liu X, Zhan P. Wang X, et al. Among authors: gao p. Curr Med Chem. 2018;25(14):1682-1702. doi: 10.2174/0929867324666170113110839. Curr Med Chem. 2018. PMID: 28088905 Review.

8

Identification of spirocyclic or phosphate substituted quinolizine derivatives as novel HIV-1 integrase inhibitors: a patent evaluation of WO2016094197A1, WO2016094198A1 and WO2016154527A1.

Cheng X, Gao P, Sun L, Tian Y, Zhan P, Liu X. Cheng X, et al. Among authors: gao p. Expert Opin Ther Pat. 2017 Nov;27(11):1277-1286. doi: 10.1080/13543776.2017.1360283. Epub 2017 Aug 2. Expert Opin Ther Pat. 2017. PMID: 28749251 Review.

9

1-Hydroxypyrido[2,3-d]pyrimidin-2(1H)-ones as novel selective HIV integrase inhibitors obtained via privileged substructure-based compound libraries.

Gao P, Zhang L, Sun L, Huang T, Tan J, Zhang J, Zhou Z, Zhao T, Menéndez-Arias L, Pannecouque C, Clercq E, Zhan P, Liu X. Gao P, et al. Bioorg Med Chem. 2017 Oct 15;25(20):5779-5789. doi: 10.1016/j.bmc.2017.09.006. Epub 2017 Sep 8. Bioorg Med Chem. 2017. PMID: 28951095

10

Recent progress in the structural modification and pharmacological activities of ligustrazine derivatives.

Zou J, Gao P, Hao X, Xu H, Zhan P, Liu X. Zou J, et al. Among authors: gao p. Eur J Med Chem. 2018 Mar 10;147:150-162. doi: 10.1016/j.ejmech.2018.01.097. Epub 2018 Feb 5. Eur J Med Chem. 2018. PMID: 29432947 Review.

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