Hulpia F - Search Results

1

New fluoroethyl phenylalanine analogues as potential LAT1-targeting PET tracers for glioblastoma.

Verhoeven J, Hulpia F, Kersemans K, Bolcaen J, De Lombaerde S, Goeman J, Descamps B, Hallaert G, Van den Broecke C, Deblaere K, Vanhove C, Van der Eycken J, Van Calenbergh S, Goethals I, De Vos F. Verhoeven J, et al. Among authors: hulpia f. Sci Rep. 2019 Feb 27;9(1):2878. doi: 10.1038/s41598-019-40013-x. Sci Rep. 2019. PMID: 30814660 Free PMC article.

2

Exploring the purine core of 3'-C-ethynyladenosine (EAdo) in search of novel nucleoside therapeutics.

Hulpia F, Balzarini J, Schols D, Andrei G, Snoeck R, Van Calenbergh S. Hulpia F, et al. Bioorg Med Chem Lett. 2016 Apr 15;26(8):1970-2. doi: 10.1016/j.bmcl.2016.03.005. Epub 2016 Mar 3. Bioorg Med Chem Lett. 2016. PMID: 26965865 Free PMC article.

3

Synthesis, in vitro and in vivo small-animal SPECT evaluation of novel technetium labeled bile acid analogues to study (altered) hepatic transporter function.

Neyt S, Vliegen M, Verreet B, De Lombaerde S, Braeckman K, Vanhove C, Huisman MT, Dumolyn C, Kersemans K, Hulpia F, Van Calenbergh S, Mannens G, De Vos F. Neyt S, et al. Among authors: hulpia f. Nucl Med Biol. 2016 Oct;43(10):642-9. doi: 10.1016/j.nucmedbio.2016.07.001. Epub 2016 Jul 12. Nucl Med Biol. 2016. PMID: 27513813

4

Synthesis of a 3'-C-ethynyl-β-d-ribofuranose purine nucleoside library: Discovery of C7-deazapurine analogs as potent antiproliferative nucleosides.

Hulpia F, Noppen S, Schols D, Andrei G, Snoeck R, Liekens S, Vervaeke P, Van Calenbergh S. Hulpia F, et al. Eur J Med Chem. 2018 Sep 5;157:248-267. doi: 10.1016/j.ejmech.2018.07.062. Epub 2018 Jul 29. Eur J Med Chem. 2018. PMID: 30098481 Free PMC article.

5

Revisiting tubercidin against kinetoplastid parasites: Aromatic substitutions at position 7 improve activity and reduce toxicity.

Hulpia F, Campagnaro GD, Scortichini M, Van Hecke K, Maes L, de Koning HP, Caljon G, Van Calenbergh S. Hulpia F, et al. Eur J Med Chem. 2019 Feb 15;164:689-705. doi: 10.1016/j.ejmech.2018.12.050. Epub 2018 Dec 21. Eur J Med Chem. 2019. PMID: 30677668

6

Discovery of Pyrrolo[2,3-b]pyridine (1,7-Dideazapurine) Nucleoside Analogues as Anti-Trypanosoma cruzi Agents.

Lin C, Hulpia F, da Silva CF, Batista DDGJ, Van Hecke K, Maes L, Caljon G, Soeiro MNC, Van Calenbergh S. Lin C, et al. Among authors: hulpia f. J Med Chem. 2019 Oct 10;62(19):8847-8865. doi: 10.1021/acs.jmedchem.9b01275. Epub 2019 Sep 20. J Med Chem. 2019. PMID: 31495177

7

Combining tubercidin and cordycepin scaffolds results in highly active candidates to treat late-stage sleeping sickness.

Hulpia F, Mabille D, Campagnaro GD, Schumann G, Maes L, Roditi I, Hofer A, de Koning HP, Caljon G, Van Calenbergh S. Hulpia F, et al. Nat Commun. 2019 Dec 5;10(1):5564. doi: 10.1038/s41467-019-13522-6. Nat Commun. 2019. PMID: 31804484 Free PMC article.

8

C6-O-alkylated 7-deazainosine nucleoside analogues: Discovery of potent and selective anti-sleeping sickness agents.

Hulpia F, Bouton J, Campagnaro GD, Alfayez IA, Mabille D, Maes L, de Koning HP, Caljon G, Van Calenbergh S. Hulpia F, et al. Eur J Med Chem. 2020 Feb 15;188:112018. doi: 10.1016/j.ejmech.2019.112018. Epub 2020 Jan 3. Eur J Med Chem. 2020. PMID: 31931339 Free article.

9

1-(1-Arylethylpiperidin-4-yl)thymine Analogs as Antimycobacterial TMPK Inhibitors.

Jian Y, Hulpia F, D P Risseeuw M, Forbes HE, Caljon G, Munier-Lehmann H, I M Boshoff H, Van Calenbergh S. Jian Y, et al. Among authors: hulpia f. Molecules. 2020 Jun 17;25(12):2805. doi: 10.3390/molecules25122805. Molecules. 2020. PMID: 32560578 Free PMC article.

10

Synthesis and structure activity relationships of cyanopyridone based anti-tuberculosis agents.

Jian Y, Hulpia F, Risseeuw MDP, Forbes HE, Munier-Lehmann H, Caljon G, Boshoff HIM, Van Calenbergh S. Jian Y, et al. Among authors: hulpia f. Eur J Med Chem. 2020 Sep 1;201:112450. doi: 10.1016/j.ejmech.2020.112450. Epub 2020 Jun 12. Eur J Med Chem. 2020. PMID: 32623208 Free PMC article.

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