Contini A - Search Results

1

Identification of the first enantiopure Rac1-Tiam1 protein-protein interaction inhibitor and its optimized synthesis via phosphine free remote group directed hydroarylation.

Ruffoni A, Ferri N, Pinto A, Pellegrino S, Contini A, Clerici F. Ruffoni A, et al. Among authors: contini a. Medchemcomm. 2018 Dec 26;10(2):310-314. doi: 10.1039/c8md00477c. eCollection 2019 Feb 1. Medchemcomm. 2018. PMID: 30931091 Free PMC article.

2

Isothiazoles. Part XV. A mild and efficient synthesis of new antiproliferative 5-sulfanylsubstituted 3-alkylaminoisothiazole 1,1-dioxides.

Clerici F, Contini A, Corsini A, Ferri N, Grzesiak S, Pellegrino S, Sala A, Yokoyama K. Clerici F, et al. Among authors: contini a. Eur J Med Chem. 2006 May;41(5):675-82. doi: 10.1016/j.ejmech.2006.01.009. Epub 2006 Mar 15. Eur J Med Chem. 2006. PMID: 16540206

3

Virtual screening approach for the identification of new Rac1 inhibitors.

Ferri N, Corsini A, Bottino P, Clerici F, Contini A. Ferri N, et al. Among authors: contini a. J Med Chem. 2009 Jul 23;52(14):4087-90. doi: 10.1021/jm8015987. J Med Chem. 2009. PMID: 19527032

4

A highly diastereoselective synthesis of α-hydroxy-β-amino acid derivatives via a Lewis acid catalyzed three-component condensation reaction.

Gassa F, Contini A, Fontana G, Pellegrino S, Gelmi ML. Gassa F, et al. Among authors: contini a. J Org Chem. 2010 Nov 5;75(21):7099-106. doi: 10.1021/jo1011762. J Org Chem. 2010. PMID: 20945864

5

Synthesis, structural, and biological evaluation of bis-heteroarylmaleimides and bis-heterofused imides.

Ferri N, Radice T, Antonino M, Beccalli EM, Tinelli S, Zunino F, Corsini A, Pratesi G, Ragg EM, Gelmi ML, Contini A. Ferri N, et al. Among authors: contini a. Bioorg Med Chem. 2011 Sep 15;19(18):5291-9. doi: 10.1016/j.bmc.2011.08.016. Epub 2011 Aug 16. Bioorg Med Chem. 2011. PMID: 21880496

6

Expedient chemical synthesis of 75mer DNA binding domain of MafA: an insight on its binding to insulin enhancer.

Pellegrino S, Annoni C, Contini A, Clerici F, Gelmi ML. Pellegrino S, et al. Among authors: contini a. Amino Acids. 2012 Nov;43(5):1995-2003. doi: 10.1007/s00726-012-1274-2. Epub 2012 Apr 4. Amino Acids. 2012. PMID: 22476346

7

1H-Azepine-4-amino-4-carboxylic acid: a new α,α-disubstituted ornithine analogue capable of inducing helix conformations in short Ala-Aib pentapeptides.

Pellegrino S, Contini A, Clerici F, Gori A, Nava D, Gelmi ML. Pellegrino S, et al. Among authors: contini a. Chemistry. 2012 Jul 9;18(28):8705-15. doi: 10.1002/chem.201104023. Epub 2012 Jun 11. Chemistry. 2012. PMID: 22689465

8

Molecular dynamic simulation of mGluR5 amino terminal domain: essential dynamics analysis captures the agonist or antagonist behaviour of ligands.

Casoni A, Clerici F, Contini A. Casoni A, et al. Among authors: contini a. J Mol Graph Model. 2013 Apr;41:72-8. doi: 10.1016/j.jmgm.2013.02.002. Epub 2013 Feb 14. J Mol Graph Model. 2013. PMID: 23500630 Free article.

9

Role of small GTPase protein Rac1 in cardiovascular diseases: development of new selective pharmacological inhibitors.

Ferri N, Contini A, Bernini SK, Corsini A. Ferri N, et al. Among authors: contini a. J Cardiovasc Pharmacol. 2013 Nov;62(5):425-35. doi: 10.1097/FJC.0b013e3182a18bcc. J Cardiovasc Pharmacol. 2013. PMID: 23921306 Review.

10

2-Amino-3-(phenylsulfanyl)norbornane-2-carboxylate: an appealing scaffold for the design of Rac1-Tiam1 protein-protein interaction inhibitors.

Ruffoni A, Ferri N, Bernini SK, Ricci C, Corsini A, Maffucci I, Clerici F, Contini A. Ruffoni A, et al. Among authors: contini a. J Med Chem. 2014 Apr 10;57(7):2953-62. doi: 10.1021/jm401924s. Epub 2014 Feb 21. J Med Chem. 2014. PMID: 24520998

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