Krasavin M - Search Results

1

1,2,4-Oxadiazole/2-Imidazoline Hybrids: Multi-target-directed Compounds for the Treatment of Infectious Diseases and Cancer.

Shetnev A, Baykov S, Kalinin S, Belova A, Sharoyko V, Rozhkov A, Zelenkov L, Tarasenko M, Sadykov E, Korsakov M, Krasavin M. Shetnev A, et al. Among authors: krasavin m. Int J Mol Sci. 2019 Apr 5;20(7):1699. doi: 10.3390/ijms20071699. Int J Mol Sci. 2019. PMID: 30959765 Free PMC article.

2

Probing the 'bipolar' nature of the carbonic anhydrase active site: aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms.

Krasavin M, Korsakov M, Dorogov M, Tuccinardi T, Dedeoglu N, Supuran CT. Krasavin M, et al. Eur J Med Chem. 2015 Aug 28;101:334-47. doi: 10.1016/j.ejmech.2015.06.022. Epub 2015 Jun 25. Eur J Med Chem. 2015. PMID: 26160114

3

Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases.

Supuran CT, Kalinin S, Tanç M, Sarnpitak P, Mujumdar P, Poulsen SA, Krasavin M. Supuran CT, et al. Among authors: krasavin m. J Enzyme Inhib Med Chem. 2016;31(sup1):197-202. doi: 10.1080/14756366.2016.1178248. Epub 2016 May 10. J Enzyme Inhib Med Chem. 2016. PMID: 27160030 Free article.

4

Multicomponent chemistry in the synthesis of carbonic anhydrase inhibitors.

Kalinin S, Supuran CT, Krasavin M. Kalinin S, et al. Among authors: krasavin m. J Enzyme Inhib Med Chem. 2016;31(sup4):185-199. doi: 10.1080/14756366.2016.1220944. Epub 2016 Oct 26. J Enzyme Inhib Med Chem. 2016. PMID: 27784162 Free article. Review.

5

Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds.

Krasavin M, Korsakov M, Zvonaryova Z, Semyonychev E, Tuccinardi T, Kalinin S, Tanç M, Supuran CT. Krasavin M, et al. Bioorg Med Chem. 2017 Mar 15;25(6):1914-1925. doi: 10.1016/j.bmc.2017.02.018. Epub 2017 Feb 13. Bioorg Med Chem. 2017. PMID: 28237553

6

Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases.

Krasavin M, Korsakov M, Ronzhina O, Tuccinardi T, Kalinin S, Tanç M, Supuran CT. Krasavin M, et al. J Enzyme Inhib Med Chem. 2017 Dec;32(1):920-934. doi: 10.1080/14756366.2017.1344236. J Enzyme Inhib Med Chem. 2017. PMID: 28718328 Free PMC article.

7

1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads.

Ferraroni M, Lucarini L, Masini E, Korsakov M, Scozzafava A, Supuran CT, Krasavin M. Ferraroni M, et al. Among authors: krasavin m. Bioorg Med Chem. 2017 Sep 1;25(17):4560-4565. doi: 10.1016/j.bmc.2017.06.054. Epub 2017 Jul 11. Bioorg Med Chem. 2017. PMID: 28728897

8

Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII.

Kalinin S, Kopylov S, Tuccinardi T, Sapegin A, Dar'in D, Angeli A, Supuran CT, Krasavin M. Kalinin S, et al. Among authors: krasavin m. ACS Med Chem Lett. 2017 Sep 15;8(10):1105-1109. doi: 10.1021/acsmedchemlett.7b00300. eCollection 2017 Oct 12. ACS Med Chem Lett. 2017. PMID: 29057059 Free PMC article.

9

Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms.

Krasavin M, Shetnev A, Sharonova T, Baykov S, Tuccinardi T, Kalinin S, Angeli A, Supuran CT. Krasavin M, et al. Bioorg Chem. 2018 Feb;76:88-97. doi: 10.1016/j.bioorg.2017.10.005. Epub 2017 Oct 16. Bioorg Chem. 2018. PMID: 29153590

10

Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors.

Sapegin A, Kalinin S, Angeli A, Supuran CT, Krasavin M. Sapegin A, et al. Among authors: krasavin m. Bioorg Chem. 2018 Feb;76:140-146. doi: 10.1016/j.bioorg.2017.11.014. Epub 2017 Nov 21. Bioorg Chem. 2018. PMID: 29175585

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