Tondi D - Search Results

1

X-ray Crystallography Deciphers the Activity of Broad-Spectrum Boronic Acid β-Lactamase Inhibitors.

Cendron L, Quotadamo A, Maso L, Bellio P, Montanari M, Celenza G, Venturelli A, Costi MP, Tondi D. Cendron L, et al. Among authors: tondi d. ACS Med Chem Lett. 2019 Mar 27;10(4):650-655. doi: 10.1021/acsmedchemlett.8b00607. eCollection 2019 Apr 11. ACS Med Chem Lett. 2019. PMID: 30996812 Free PMC article.

2

Conformational analysis of phthalein derivatives acting as thymidylate synthase inhibitors by means of 1H NMR and quantum chemical calculations.

Ghelli S, Rastelli G, Barlocco D, Rinaldi M, Tondi D, Pecorari P, Costi MP. Ghelli S, et al. Among authors: tondi d. Bioorg Med Chem. 1996 Oct;4(10):1783-94. doi: 10.1016/0968-0896(96)00193-9. Bioorg Med Chem. 1996. PMID: 8931948

3

Structure-based discovery and in-parallel optimization of novel competitive inhibitors of thymidylate synthase.

Tondi D, Slomczynska U, Costi MP, Watterson DM, Ghelli S, Shoichet BK. Tondi D, et al. Chem Biol. 1999 May;6(5):319-31. doi: 10.1016/S1074-5521(99)80077-5. Chem Biol. 1999. PMID: 10322126

4

Structure-based design and in-parallel synthesis of inhibitors of AmpC beta-lactamase.

Tondi D, Powers RA, Caselli E, Negri MC, Blázquez J, Costi MP, Shoichet BK. Tondi D, et al. Chem Biol. 2001 Jun;8(6):593-611. doi: 10.1016/s1074-5521(01)00034-5. Chem Biol. 2001. PMID: 11410378

5

Predicting and harnessing protein flexibility in the design of species-specific inhibitors of thymidylate synthase.

Fritz TA, Tondi D, Finer-Moore JS, Costi MP, Stroud RM. Fritz TA, et al. Among authors: tondi d. Chem Biol. 2001 Oct;8(10):981-95. doi: 10.1016/s1074-5521(01)00067-9. Chem Biol. 2001. PMID: 11590022

6

Structure-based studies on species-specific inhibition of thymidylate synthase.

Costi MP, Tondi D, Rinaldi M, Barlocco D, Pecorari P, Soragni F, Venturelli A, Stroud RM. Costi MP, et al. Among authors: tondi d. Biochim Biophys Acta. 2002 Jul 18;1587(2-3):206-14. doi: 10.1016/s0925-4439(02)00083-2. Biochim Biophys Acta. 2002. PMID: 12084462 Free article. Review.

7

ortho-Halogen naphthaleins as specific inhibitors of Lactobacillus casei thymidylate synthase. Conformational properties and biological activity.

Ghelli S, Rinaldi M, Barlocco D, Gelain A, Pecorari P, Tondi D, Rastelli G, Costi MP. Ghelli S, et al. Among authors: tondi d. Bioorg Med Chem. 2003 Mar 20;11(6):951-63. doi: 10.1016/s0968-0896(02)00541-2. Bioorg Med Chem. 2003. PMID: 12614880

8

Improving specificity vs bacterial thymidylate synthases through N-dansyl modulation of didansyltyrosine.

Tondi D, Venturelli A, Ferrari S, Ghelli S, Costi MP. Tondi D, et al. J Med Chem. 2005 Feb 24;48(4):913-6. doi: 10.1021/jm0491445. J Med Chem. 2005. PMID: 15715461

9

Structure-based optimization of a non-beta-lactam lead results in inhibitors that do not up-regulate beta-lactamase expression in cell culture.

Tondi D, Morandi F, Bonnet R, Costi MP, Shoichet BK. Tondi D, et al. J Am Chem Soc. 2005 Apr 6;127(13):4632-9. doi: 10.1021/ja042984o. J Am Chem Soc. 2005. PMID: 15796528 Free PMC article.

10

Thymidylate synthase structure, function and implication in drug discovery.

Costi MP, Ferrari S, Venturelli A, Calò S, Tondi D, Barlocco D. Costi MP, et al. Among authors: tondi d. Curr Med Chem. 2005;12(19):2241-58. doi: 10.2174/0929867054864868. Curr Med Chem. 2005. PMID: 16178783 Review.

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