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Page 1
Heteroaromatic rings of the future.
Pitt WR, Parry DM, Perry BG, Groom CR. Pitt WR, et al. J Med Chem. 2009 May 14;52(9):2952-63. doi: 10.1021/jm801513z. J Med Chem. 2009. PMID: 19348472
Discovery of a Potent, Orally Bioavailable PI4KIIIβ Inhibitor (UCB9608) Able To Significantly Prolong Allogeneic Organ Engraftment in Vivo.
Reuberson J, Horsley H, Franklin RJ, Ford D, Neuss J, Brookings D, Huang Q, Vanderhoydonck B, Gao LJ, Jang MY, Herdewijn P, Ghawalkar A, Fallah-Arani F, Khan AR, Henshall J, Jairaj M, Malcolm S, Ward E, Shuttleworth L, Lin Y, Li S, Louat T, Waer M, Herman J, Payne A, Ceska T, Doyle C, Pitt W, Calmiano M, Augustin M, Steinbacher S, Lammens A, Allen R. Reuberson J, et al. J Med Chem. 2018 Aug 9;61(15):6705-6723. doi: 10.1021/acs.jmedchem.8b00521. Epub 2018 Jul 19. J Med Chem. 2018. PMID: 29952567
Real-World Applications and Experiences of AI/ML Deployment for Drug Discovery.
Pitt WR, Bentley J, Boldron C, Colliandre L, Esposito C, Frush EH, Kopec J, Labouille S, Meneyrol J, Pardoe DA, Palazzesi F, Pozzan A, Remington JM, Rex R, Southey M, Vishwakarma S, Walker P. Pitt WR, et al. J Med Chem. 2025 Jan 8. doi: 10.1021/acs.jmedchem.4c03044. Online ahead of print. J Med Chem. 2025. PMID: 39772505 No abstract available.
A novel series of potent and selective IKK2 inhibitors.
Bingham AH, Davenport RJ, Gowers L, Knight RL, Lowe C, Owen DA, Parry DM, Pitt WR. Bingham AH, et al. Among authors: pitt wr. Bioorg Med Chem Lett. 2004 Jan 19;14(2):409-12. doi: 10.1016/j.bmcl.2003.10.047. Bioorg Med Chem Lett. 2004. PMID: 14698170
Novel 7-methoxy-6-oxazol-5-yl-2,3-dihydro-1H-quinazolin-4-ones as IMPDH inhibitors.
Birch HL, Buckley GM, Davies N, Dyke HJ, Frost EJ, Gilbert PJ, Hannah DR, Haughan AF, Madigan MJ, Morgan T, Pitt WR, Ratcliffe AJ, Ray NC, Richard MD, Sharpe A, Taylor AJ, Whitworth JM, Williams SC. Birch HL, et al. Among authors: pitt wr. Bioorg Med Chem Lett. 2005 Dec 1;15(23):5335-9. doi: 10.1016/j.bmcl.2005.06.108. Epub 2005 Oct 3. Bioorg Med Chem Lett. 2005. PMID: 16202581
57 results