Kalinin S - Search Results

1

Highly hydrophilic 1,3-oxazol-5-yl benzenesulfonamide inhibitors of carbonic anhydrase II for reduction of glaucoma-related intraocular pressure.

Kalinin S, Valtari A, Ruponen M, Toropainen E, Kovalenko A, Nocentini A, Gureev M, Dar'in D, Urtti A, Supuran CT, Krasavin M. Kalinin S, et al. Bioorg Med Chem. 2019 Nov 1;27(21):115086. doi: 10.1016/j.bmc.2019.115086. Epub 2019 Sep 4. Bioorg Med Chem. 2019. PMID: 31515057

2

Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases.

Supuran CT, Kalinin S, Tanç M, Sarnpitak P, Mujumdar P, Poulsen SA, Krasavin M. Supuran CT, et al. Among authors: kalinin s. J Enzyme Inhib Med Chem. 2016;31(sup1):197-202. doi: 10.1080/14756366.2016.1178248. Epub 2016 May 10. J Enzyme Inhib Med Chem. 2016. PMID: 27160030 Free article.

3

Multicomponent chemistry in the synthesis of carbonic anhydrase inhibitors.

Kalinin S, Supuran CT, Krasavin M. Kalinin S, et al. J Enzyme Inhib Med Chem. 2016;31(sup4):185-199. doi: 10.1080/14756366.2016.1220944. Epub 2016 Oct 26. J Enzyme Inhib Med Chem. 2016. PMID: 27784162 Free article. Review.

4

Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds.

Krasavin M, Korsakov M, Zvonaryova Z, Semyonychev E, Tuccinardi T, Kalinin S, Tanç M, Supuran CT. Krasavin M, et al. Among authors: kalinin s. Bioorg Med Chem. 2017 Mar 15;25(6):1914-1925. doi: 10.1016/j.bmc.2017.02.018. Epub 2017 Feb 13. Bioorg Med Chem. 2017. PMID: 28237553

5

Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases.

Krasavin M, Korsakov M, Ronzhina O, Tuccinardi T, Kalinin S, Tanç M, Supuran CT. Krasavin M, et al. Among authors: kalinin s. J Enzyme Inhib Med Chem. 2017 Dec;32(1):920-934. doi: 10.1080/14756366.2017.1344236. J Enzyme Inhib Med Chem. 2017. PMID: 28718328 Free PMC article.

6

Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII.

Kalinin S, Kopylov S, Tuccinardi T, Sapegin A, Dar'in D, Angeli A, Supuran CT, Krasavin M. Kalinin S, et al. ACS Med Chem Lett. 2017 Sep 15;8(10):1105-1109. doi: 10.1021/acsmedchemlett.7b00300. eCollection 2017 Oct 12. ACS Med Chem Lett. 2017. PMID: 29057059 Free PMC article.

7

Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms.

Krasavin M, Shetnev A, Sharonova T, Baykov S, Tuccinardi T, Kalinin S, Angeli A, Supuran CT. Krasavin M, et al. Among authors: kalinin s. Bioorg Chem. 2018 Feb;76:88-97. doi: 10.1016/j.bioorg.2017.10.005. Epub 2017 Oct 16. Bioorg Chem. 2018. PMID: 29153590

8

Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors.

Sapegin A, Kalinin S, Angeli A, Supuran CT, Krasavin M. Sapegin A, et al. Among authors: kalinin s. Bioorg Chem. 2018 Feb;76:140-146. doi: 10.1016/j.bioorg.2017.11.014. Epub 2017 Nov 21. Bioorg Chem. 2018. PMID: 29175585

9

Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment.

Krasavin M, Shetnev A, Sharonova T, Baykov S, Kalinin S, Nocentini A, Sharoyko V, Poli G, Tuccinardi T, Presnukhina S, Tennikova TB, Supuran CT. Krasavin M, et al. Among authors: kalinin s. Eur J Med Chem. 2019 Feb 15;164:92-105. doi: 10.1016/j.ejmech.2018.12.049. Epub 2018 Dec 21. Eur J Med Chem. 2019. PMID: 30594030

10

Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines.

Krasavin M, Shetnev A, Baykov S, Kalinin S, Nocentini A, Sharoyko V, Poli G, Tuccinardi T, Korsakov M, Tennikova TB, Supuran CT. Krasavin M, et al. Among authors: kalinin s. Eur J Med Chem. 2019 Apr 15;168:301-314. doi: 10.1016/j.ejmech.2019.02.044. Epub 2019 Feb 15. Eur J Med Chem. 2019. PMID: 30826507

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