Hirasawa A - Search Results

1

Structural insights for producing CK2α1-specific inhibitors.

Tsuyuguchi M, Nakaniwa T, Hirasawa A, Nakanishi I, Kinoshita T. Tsuyuguchi M, et al. Among authors: hirasawa a. Bioorg Med Chem Lett. 2020 Jan 15;30(2):126837. doi: 10.1016/j.bmcl.2019.126837. Epub 2019 Dec 3. Bioorg Med Chem Lett. 2020. PMID: 31859160

2

Structure-activity relationships of pyrazine-based CK2 inhibitors: synthesis and evaluation of 2,6-disubstituted pyrazines and 4,6-disubstituted pyrimidines.

Suzuki Y, Cluzeau J, Hara T, Hirasawa A, Tsujimoto G, Oishi S, Ohno H, Fujii N. Suzuki Y, et al. Among authors: hirasawa a. Arch Pharm (Weinheim). 2008 Sep;341(9):554-61. doi: 10.1002/ardp.200700269. Arch Pharm (Weinheim). 2008. PMID: 18763715

3

Structure of human protein kinase CK2 alpha 2 with a potent indazole-derivative inhibitor.

Nakaniwa T, Kinoshita T, Sekiguchi Y, Tada T, Nakanishi I, Kitaura K, Suzuki Y, Ohno H, Hirasawa A, Tsujimoto G. Nakaniwa T, et al. Among authors: hirasawa a. Acta Crystallogr Sect F Struct Biol Cryst Commun. 2009 Feb 1;65(Pt 2):75-9. doi: 10.1107/S1744309108043194. Epub 2009 Jan 31. Acta Crystallogr Sect F Struct Biol Cryst Commun. 2009. PMID: 19193990 Free PMC article.

4

Structural insight into human CK2alpha in complex with the potent inhibitor ellagic acid.

Sekiguchi Y, Nakaniwa T, Kinoshita T, Nakanishi I, Kitaura K, Hirasawa A, Tsujimoto G, Tada T. Sekiguchi Y, et al. Among authors: hirasawa a. Bioorg Med Chem Lett. 2009 Jun 1;19(11):2920-3. doi: 10.1016/j.bmcl.2009.04.076. Epub 2009 Apr 22. Bioorg Med Chem Lett. 2009. PMID: 19414254

5

A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase.

Kinoshita T, Sekiguchi Y, Fukada H, Nakaniwa T, Tada T, Nakamura S, Kitaura K, Ohno H, Suzuki Y, Hirasawa A, Nakanishi I, Tsujimoto G. Kinoshita T, et al. Among authors: hirasawa a. Mol Cell Biochem. 2011 Oct;356(1-2):97-105. doi: 10.1007/s11010-011-0960-9. Epub 2011 Jul 7. Mol Cell Biochem. 2011. PMID: 21735094

6

Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds.

Hou Z, Nakanishi I, Kinoshita T, Takei Y, Yasue M, Misu R, Suzuki Y, Nakamura S, Kure T, Ohno H, Murata K, Kitaura K, Hirasawa A, Tsujimoto G, Oishi S, Fujii N. Hou Z, et al. Among authors: hirasawa a. J Med Chem. 2012 Mar 22;55(6):2899-903. doi: 10.1021/jm2015167. Epub 2012 Mar 7. J Med Chem. 2012. PMID: 22339433

7

Design and synthesis of a novel class of CK2 inhibitors: application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles.

Suzuki Y, Oishi S, Takei Y, Yasue M, Misu R, Naoe S, Hou Z, Kure T, Nakanishi I, Ohno H, Hirasawa A, Tsujimoto G, Fujii N. Suzuki Y, et al. Among authors: hirasawa a. Org Biomol Chem. 2012 Jul 7;10(25):4907-15. doi: 10.1039/c2ob25298h. Epub 2012 May 21. Org Biomol Chem. 2012. PMID: 22610034 Free article.

8

Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: application to the development of a new class of CK2 inhibitors.

Hou Z, Oishi S, Suzuki Y, Kure T, Nakanishi I, Hirasawa A, Tsujimoto G, Ohno H, Fujii N. Hou Z, et al. Among authors: hirasawa a. Org Biomol Chem. 2013 May 28;11(20):3288-96. doi: 10.1039/c3ob40223a. Org Biomol Chem. 2013. PMID: 23535832 Free article.

9

Identification of protein kinase CK2 inhibitors using solvent dipole ordering virtual screening.

Nakanishi I, Murata K, Nagata N, Kurono M, Kinoshita T, Yasue M, Miyazaki T, Takei Y, Nakamura S, Sakurai A, Iwamoto N, Nishiwaki K, Nakaniwa T, Sekiguchi Y, Hirasawa A, Tsujimoto G, Kitaura K. Nakanishi I, et al. Among authors: hirasawa a. Eur J Med Chem. 2015;96:396-404. doi: 10.1016/j.ejmech.2015.04.032. Epub 2015 Apr 15. Eur J Med Chem. 2015. PMID: 25912672

10

Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists.

Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Navenot JM, Peiper SC, Fujii N. Masuda R, et al. Among authors: hirasawa a. Bioconjug Chem. 2012 Jun 20;23(6):1259-65. doi: 10.1021/bc300084h. Epub 2012 May 9. Bioconjug Chem. 2012. PMID: 22486464

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