Sors A - Search Results

1

Safety and efficacy of GABA_A α5 antagonist S44819 in patients with ischaemic stroke: a multicentre, double-blind, randomised, placebo-controlled trial.

Chabriat H, Bassetti CL, Marx U, Audoli-Inthavong ML, Sors A, Lambert E, Wattez M, Hermann DM; RESTORE BRAIN study investigators. Chabriat H, et al. Among authors: sors a. Lancet Neurol. 2020 Mar;19(3):226-233. doi: 10.1016/S1474-4422(20)30004-1. Lancet Neurol. 2020. PMID: 32085836 Clinical Trial.

2

Randomized Efficacy and Safety Trial with Oral S 44819 after Recent ischemic cerebral Event (RESTORE BRAIN study): a placebo controlled phase II study.

Chabriat H, Bassetti CL, Marx U, Picarel-Blanchot F, Sors A, Gruget C, Saba B, Wattez M, Audoli ML, Hermann DM. Chabriat H, et al. Among authors: sors a. Trials. 2020 Feb 3;21(1):136. doi: 10.1186/s13063-020-4072-2. Trials. 2020. PMID: 32014032 Free PMC article. Clinical Trial.

3

Preclinical concepts and results with the GABA_A antagonist S44819 in a mouse model of middle cerebral artery occlusion.

Hermann DM, Saba B, Sors A, Bassetti CL. Hermann DM, et al. Among authors: sors a. Neural Regen Res. 2019 Sep;14(9):1517-1518. doi: 10.4103/1673-5374.255963. Neural Regen Res. 2019. PMID: 31089046 Free PMC article. No abstract available.

4

Post-acute delivery of α5-GABAA antagonist, S 44819, improves functional recovery in juvenile rats following stroke.

Lebrun F, Violle N, Letourneur A, Muller C, Fischer N, Levilly A, Orset C, Sors A, Vivien D. Lebrun F, et al. Among authors: sors a. Exp Neurol. 2022 Jan;347:113881. doi: 10.1016/j.expneurol.2021.113881. Epub 2021 Sep 29. Exp Neurol. 2022. PMID: 34597681

5

Effects of S 38093, an antagonist/inverse agonist of histamine H3 receptors, in models of neuropathic pain in rats.

Chaumette T, Chapuy E, Berrocoso E, Llorca-Torralba M, Bravo L, Mico JA, Chalus M, Eschalier A, Ardid D, Marchand F, Sors A. Chaumette T, et al. Among authors: sors a. Eur J Pain. 2018 Jan;22(1):127-141. doi: 10.1002/ejp.1097. Epub 2017 Sep 6. Eur J Pain. 2018. PMID: 28877402

6

Mechanistic characterization of S 38093, a novel inverse agonist at histamine H3 receptors.

Sors A, Panayi F, Bert L, Favale D, Nosjean O, Audinot V, Arrang JM, Buisson B, Steidl E, Delbos JM, Huhtala T, Kontkanen O, Chollet AM, Casara P, Lestage P. Sors A, et al. Eur J Pharmacol. 2017 May 15;803:11-23. doi: 10.1016/j.ejphar.2017.03.013. Epub 2017 Mar 21. Eur J Pharmacol. 2017. PMID: 28336400

7

In vivo pharmacological profile of S 38093, a novel histamine H3 receptor inverse agonist.

Panayi F, Sors A, Bert L, Martin B, Rollin-Jego G, Billiras R, Carrié I, Albinet K, Danober L, Rogez N, Thomas JY, Pira L, Bertaina-Anglade V, Lestage P. Panayi F, et al. Among authors: sors a. Eur J Pharmacol. 2017 May 15;803:1-10. doi: 10.1016/j.ejphar.2017.03.008. Epub 2017 Mar 14. Eur J Pharmacol. 2017. PMID: 28315340

8

Drug-receptor kinetics and sigma-1 receptor affinity differentiate clinically evaluated histamine H₃ receptor antagonists.

Riddy DM, Cook AE, Shackleford DM, Pierce TL, Mocaer E, Mannoury la Cour C, Sors A, Charman WN, Summers RJ, Sexton PM, Christopoulos A, Langmead CJ. Riddy DM, et al. Among authors: sors a. Neuropharmacology. 2019 Jan;144:244-255. doi: 10.1016/j.neuropharm.2018.10.028. Epub 2018 Oct 22. Neuropharmacology. 2019. PMID: 30359639

9

S 38093, a histamine H₃ antagonist/inverse agonist, promotes hippocampal neurogenesis and improves context discrimination task in aged mice.

Guilloux JP, Samuels BA, Mendez-David I, Hu A, Levinstein M, Faye C, Mekiri M, Mocaer E, Gardier AM, Hen R, Sors A, David DJ. Guilloux JP, et al. Among authors: sors a. Sci Rep. 2017 Feb 20;7:42946. doi: 10.1038/srep42946. Sci Rep. 2017. PMID: 28218311 Free PMC article.

10

The Synergistic Enhancing-Memory Effect of Donepezil and S 38093 (a Histamine H₃ Antagonist) Is Mediated by Increased Neural Activity in the Septo-hippocampal Circuitry in Middle-Aged Mice.

Sors A, Krazem A, Kehr J, Yoshitake T, Dominguez G, Henkous N, Letondor C, Mocaer E, Béracochéa DJ. Sors A, et al. Front Pharmacol. 2016 Dec 22;7:492. doi: 10.3389/fphar.2016.00492. eCollection 2016. Front Pharmacol. 2016. PMID: 28066242 Free PMC article.

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