Thacker PS - Search Results

1

Synthesis and biological evaluation of some coumarin hybrids as selective carbonic anhydrase IX and XII inhibitors.

Thacker PS, Sridhar Goud N, Argulwar OS, Soman J, Angeli A, Alvala M, Arifuddin M, Supuran CT. Thacker PS, et al. Bioorg Chem. 2020 Nov;104:104272. doi: 10.1016/j.bioorg.2020.104272. Epub 2020 Sep 8. Bioorg Chem. 2020. PMID: 32961467

2

Design, synthesis and biological evaluation of coumarin-3-carboxamides as selective carbonic anhydrase IX and XII inhibitors.

Thacker PS, Alvala M, Arifuddin M, Angeli A, Supuran CT. Thacker PS, et al. Bioorg Chem. 2019 May;86:386-392. doi: 10.1016/j.bioorg.2019.02.004. Epub 2019 Feb 5. Bioorg Chem. 2019. PMID: 30763885

3

Synthesis and biological evaluation of novel 8-substituted quinoline-2-carboxamides as carbonic anhydrase inhibitors.

Thacker PS, Shaikh P, Angeli A, Arifuddin M, Supuran CT. Thacker PS, et al. J Enzyme Inhib Med Chem. 2019 Dec;34(1):1172-1177. doi: 10.1080/14756366.2019.1626376. J Enzyme Inhib Med Chem. 2019. PMID: 31218888 Free PMC article.

4

Synthesis of a new series of 3-functionalised-1-phenyl-1,2,3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors.

Swain B, Angeli A, Angapelly S, Thacker PS, Singh P, Supuran CT, Arifuddin M. Swain B, et al. Among authors: thacker ps. J Enzyme Inhib Med Chem. 2019 Dec;34(1):1199-1209. doi: 10.1080/14756366.2019.1629432. J Enzyme Inhib Med Chem. 2019. PMID: 31237458 Free PMC article.

5

Design, synthesis and biological evaluation of coumarin linked 1,2,4-oxadiazoles as selective carbonic anhydrase IX and XII inhibitors.

Thacker PS, Angeli A, Argulwar OS, Tiwari PL, Arifuddin M, Supuran CT. Thacker PS, et al. Bioorg Chem. 2020 May;98:103739. doi: 10.1016/j.bioorg.2020.103739. Epub 2020 Mar 10. Bioorg Chem. 2020. PMID: 32193032

6

Synthesis and carbonic anhydrase inhibition studies of sulfonamide based indole-1,2,3-triazole chalcone hybrids.

Singh P, Swain B, Thacker PS, Sigalapalli DK, Purnachander Yadav P, Angeli A, Supuran CT, Arifuddin M. Singh P, et al. Among authors: thacker ps. Bioorg Chem. 2020 Jun;99:103839. doi: 10.1016/j.bioorg.2020.103839. Epub 2020 Apr 8. Bioorg Chem. 2020. PMID: 32289586

7

Design, Synthesis, and Biological Evaluation of 1,2,3-Triazole-Linked Triazino[5,6-B]Indole-Benzene Sulfonamide Conjugates as Potent Carbonic Anhydrase I, II, IX, and XIII Inhibitors.

Chinchilli KK, Angeli A, Thacker PS, Korra LN, Biswas R, Arifuddin M, Supuran CT. Chinchilli KK, et al. Among authors: thacker ps. Metabolites. 2020 May 15;10(5):200. doi: 10.3390/metabo10050200. Metabolites. 2020. PMID: 32429261 Free PMC article.

8

Development of quinoline-based hybrid as inhibitor of methionine aminopeptidase 1 from Leishmania donovani.

Bhat SY, Bhandari S, Thacker PS, Arifuddin M, Qureshi IA. Bhat SY, et al. Among authors: thacker ps. Chem Biol Drug Des. 2021 Feb;97(2):315-324. doi: 10.1111/cbdd.13783. Epub 2020 Sep 7. Chem Biol Drug Des. 2021. PMID: 32816410

9

Coumarin-Thiourea Hybrids Show Potent Carbonic Anhydrase IX and XIII Inhibitory Action.

Thacker PS, Srikanth D, Angeli A, Singh P, Chinchilli KK, Arifuddin M, Supuran CT. Thacker PS, et al. ChemMedChem. 2021 Apr 20;16(8):1252-1256. doi: 10.1002/cmdc.202000915. Epub 2021 Feb 9. ChemMedChem. 2021. PMID: 33346945

10

Discovery of a novel series of indolylchalcone-benzenesulfonamide hybrids acting as selective carbonic anhydrase II inhibitors.

Singh P, Purnachander Yadav P, Swain B, Thacker PS, Angeli A, Supuran CT, Arifuddin M. Singh P, et al. Among authors: thacker ps. Bioorg Chem. 2021 Mar;108:104647. doi: 10.1016/j.bioorg.2021.104647. Epub 2021 Jan 19. Bioorg Chem. 2021. PMID: 33530019

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