Altmann E - Search Results

1

Discovery of Potent, Highly Selective, and In Vivo Efficacious, Allosteric MALT1 Inhibitors by Iterative Scaffold Morphing.

Pissot Soldermann C, Simic O, Renatus M, Erbel P, Melkko S, Wartmann M, Bigaud M, Weiss A, McSheehy P, Endres R, Santos P, Blank J, Schuffenhauer A, Bold G, Buschmann N, Zoller T, Altmann E, Manley PW, Dix I, Buchdunger E, Scesa J, Quancard J, Schlapbach A, Bornancin F, Radimerski T, Régnier CH. Pissot Soldermann C, et al. Among authors: altmann e. J Med Chem. 2020 Dec 10;63(23):14576-14593. doi: 10.1021/acs.jmedchem.0c01245. Epub 2020 Nov 30. J Med Chem. 2020. PMID: 33252239

2

Substituted 5,7-diphenyl-pyrrolo[2,3d]pyrimidines: potent inhibitors of the tyrosine kinase c-Src.

Missbach M, Altmann E, Widler L, Susa M, Buchdunger E, Mett H, Meyer T, Green J. Missbach M, et al. Among authors: altmann e. Bioorg Med Chem Lett. 2000 May 1;10(9):945-9. doi: 10.1016/s0960-894x(00)00131-1. Bioorg Med Chem Lett. 2000. PMID: 10853665

3

7-Alkyl- and 7-cycloalkyl-5-aryl-pyrrolo[2,3-d]pyrimidines--potent inhibitors of the tyrosine kinase c-Src.

Widler L, Green J, Missbach M, Susa M, Altmann E. Widler L, et al. Among authors: altmann e. Bioorg Med Chem Lett. 2001 Mar 26;11(6):849-52. doi: 10.1016/s0960-894x(01)00079-8. Bioorg Med Chem Lett. 2001. PMID: 11277535

4

7-Pyrrolidinyl- and 7-piperidinyl-5-aryl-pyrrolo[2,3-d]pyrimidines--potent inhibitors of the tyrosine kinase c-Src.

Altmann E, Missbach M, Green J, Susa M, Wagenknecht HA, Widler L. Altmann E, et al. Bioorg Med Chem Lett. 2001 Mar 26;11(6):853-6. doi: 10.1016/s0960-894x(01)00080-4. Bioorg Med Chem Lett. 2001. PMID: 11277536

5

N(7)-substituted-5-aryl-pyrrolo[2,3-d]pyrimidines represent a versatile class of potent inhibitors of the tyrosine kinase c-Src.

Altmann E, Widler L, Missbach M. Altmann E, et al. Mini Rev Med Chem. 2002 Jun;2(3):201-8. doi: 10.2174/1389557023406188. Mini Rev Med Chem. 2002. PMID: 12370062 Review.

6

Arylaminoethyl amides as inhibitors of the cysteine protease cathepsin K-investigating P1' substituents.

Altmann E, Green J, Tintelnot-Blomley M. Altmann E, et al. Bioorg Med Chem Lett. 2003 Jun 16;13(12):1997-2001. doi: 10.1016/s0960-894x(03)00344-5. Bioorg Med Chem Lett. 2003. PMID: 12781182

7

Novel purine nitrile derived inhibitors of the cysteine protease cathepsin K.

Altmann E, Cowan-Jacob SW, Missbach M. Altmann E, et al. J Med Chem. 2004 Nov 18;47(24):5833-6. doi: 10.1021/jm0493111. J Med Chem. 2004. PMID: 15537340

8

Dipeptide nitrile inhibitors of cathepsin K.

Altmann E, Aichholz R, Betschart C, Buhl T, Green J, Lattmann R, Missbach M. Altmann E, et al. Bioorg Med Chem Lett. 2006 May 1;16(9):2549-54. doi: 10.1016/j.bmcl.2006.01.104. Epub 2006 Feb 9. Bioorg Med Chem Lett. 2006. PMID: 16480867

9

2-Cyano-pyrimidines: a new chemotype for inhibitors of the cysteine protease cathepsin K.

Altmann E, Aichholz R, Betschart C, Buhl T, Green J, Irie O, Teno N, Lattmann R, Tintelnot-Blomley M, Missbach M. Altmann E, et al. J Med Chem. 2007 Feb 22;50(4):591-4. doi: 10.1021/jm0613525. Epub 2007 Jan 27. J Med Chem. 2007. PMID: 17256925

10

1-Alkyl-4-phenyl-6-alkoxy-1H-quinazolin-2-ones: a novel series of potent calcium-sensing receptor antagonists.

Widler L, Altmann E, Beerli R, Breitenstein W, Bouhelal R, Buhl T, Gamse R, Gerspacher M, Halleux C, John MR, Lehmann H, Kalb O, Kneissel M, Missbach M, Müller IR, Reidemeister S, Renaud J, Taillardat A, Tommasi R, Weiler S, Wolf RM, Seuwen K. Widler L, et al. Among authors: altmann e. J Med Chem. 2010 Mar 11;53(5):2250-63. doi: 10.1021/jm901811v. J Med Chem. 2010. PMID: 20158186

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