Barral K - Search Results

1

Pharmacological inhibition of syntenin PDZ2 domain impairs breast cancer cell activities and exosome loading with syndecan and EpCAM cargo.

Leblanc R, Kashyap R, Barral K, Egea-Jimenez AL, Kovalskyy D, Feracci M, Garcia M, Derviaux C, Betzi S, Ghossoub R, Platonov M, Roche P, Morelli X, Hoffer L, Zimmermann P. Leblanc R, et al. Among authors: barral k. J Extracell Vesicles. 2020 Dec;10(2):e12039. doi: 10.1002/jev2.12039. Epub 2020 Dec 15. J Extracell Vesicles. 2020. PMID: 33343836 Free PMC article.

2

Optimization of a fragment linking hit toward Dengue and Zika virus NS5 methyltransferases inhibitors.

Hernandez J, Hoffer L, Coutard B, Querat G, Roche P, Morelli X, Decroly E, Barral K. Hernandez J, et al. Among authors: barral k. Eur J Med Chem. 2019 Jan 1;161:323-333. doi: 10.1016/j.ejmech.2018.09.056. Epub 2018 Oct 23. Eur J Med Chem. 2019. PMID: 30368131

3

Fragment-based drug design targeting syntenin PDZ2 domain involved in exosomal release and tumour spread.

Garcia M, Hoffer L, Leblanc R, Benmansour F, Feracci M, Derviaux C, Egea-Jimenez AL, Roche P, Zimmermann P, Morelli X, Barral K. Garcia M, et al. Among authors: barral k. Eur J Med Chem. 2021 Nov 5;223:113601. doi: 10.1016/j.ejmech.2021.113601. Epub 2021 Jun 5. Eur J Med Chem. 2021. PMID: 34153575

4

Discovery of a PDZ Domain Inhibitor Targeting the Syndecan/Syntenin Protein-Protein Interaction: A Semi-Automated "Hit Identification-to-Optimization" Approach.

Hoffer L, Garcia M, Leblanc R, Feracci M, Betzi S, Ben Yaala K, Daulat AM, Zimmermann P, Roche P, Barral K, Morelli X. Hoffer L, et al. Among authors: barral k. J Med Chem. 2023 Apr 13;66(7):4633-4658. doi: 10.1021/acs.jmedchem.2c01569. Epub 2023 Mar 20. J Med Chem. 2023. PMID: 36939673

5

In vitro screening of a FDA approved chemical library reveals potential inhibitors of SARS-CoV-2 replication.

Touret F, Gilles M, Barral K, Nougairède A, van Helden J, Decroly E, de Lamballerie X, Coutard B. Touret F, et al. Among authors: barral k. Sci Rep. 2020 Aug 4;10(1):13093. doi: 10.1038/s41598-020-70143-6. Sci Rep. 2020. PMID: 32753646 Free PMC article.

6

Synthesis and antiviral evaluation of cis-substituted cyclohexenyl and cyclohexanyl nucleosides.

Barral K, Courcambeck J, Pèpe G, Balzarini J, Neyts J, De Clercq E, Camplo M. Barral K, et al. J Med Chem. 2005 Jan 27;48(2):450-6. doi: 10.1021/jm0493966. J Med Chem. 2005. PMID: 15658858

7

Synthesis and antiviral evaluation of cyclic and acyclic 2-methyl-3-hydroxy-4-pyridinone nucleoside derivatives.

Barral K, Balzarini J, Neyts J, De Clercq E, Hider RC, Camplo M. Barral K, et al. J Med Chem. 2006 Jan 12;49(1):43-50. doi: 10.1021/jm0504306. J Med Chem. 2006. PMID: 16392791

8

Synthesis, in vitro antiviral evaluation, and stability studies of novel alpha-borano-nucleotide analogues of 9-[2-(phosphonomethoxy)ethyl]adenine and (R)-9-[2-(phosphonomethoxy)propyl]adenine.

Barral K, Priet S, Sire J, Neyts J, Balzarini J, Canard B, Alvarez K. Barral K, et al. J Med Chem. 2006 Dec 28;49(26):7799-806. doi: 10.1021/jm060030y. J Med Chem. 2006. PMID: 17181162

9

Synthesis and antiviral activity of boranophosphonate isosteres of AZT and d4T monophosphates.

Barral K, Priet S, De Michelis C, Sire J, Neyts J, Balzarini J, Canard B, Alvarez K. Barral K, et al. Eur J Med Chem. 2010 Feb;45(2):849-56. doi: 10.1016/j.ejmech.2009.11.012. Epub 2009 Nov 12. Eur J Med Chem. 2010. PMID: 19969396

10

Acyclic nucleoside thiophosphonates as potent inhibitors of HIV and HBV replication.

Barral K, Weck C, Payrot N, Roux L, Durafour C, Zoulim F, Neyts J, Balzarini J, Canard B, Priet S, Alvarez K. Barral K, et al. Eur J Med Chem. 2011 Sep;46(9):4281-8. doi: 10.1016/j.ejmech.2011.06.034. Epub 2011 Jul 1. Eur J Med Chem. 2011. PMID: 21803462 Free PMC article.

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