Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains.
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Mirguet O, et al. Among authors: jeffrey p.
J Med Chem. 2013 Oct 10;56(19):7501-15. doi: 10.1021/jm401088k. Epub 2013 Sep 25.
J Med Chem. 2013.
PMID: 24015967