Vernall AJ - Search Results

1

Development of Covalent, Clickable Probes for Adenosine A₁ and A₃ Receptors.

Trinh PNH, Chong DJW, Leach K, Hill SJ, Tyndall JDA, May LT, Vernall AJ, Gregory KJ. Trinh PNH, et al. Among authors: vernall aj. J Med Chem. 2021 Jun 24;64(12):8161-8178. doi: 10.1021/acs.jmedchem.0c02169. Epub 2021 Jun 14. J Med Chem. 2021. PMID: 34120444

2

Highly potent and selective fluorescent antagonists of the human adenosine A₃ receptor based on the 1,2,4-triazolo[4,3-a]quinoxalin-1-one scaffold.

Vernall AJ, Stoddart LA, Briddon SJ, Hill SJ, Kellam B. Vernall AJ, et al. J Med Chem. 2012 Feb 23;55(4):1771-82. doi: 10.1021/jm201722y. Epub 2012 Feb 13. J Med Chem. 2012. PMID: 22277057

3

Fragment screening at adenosine-A(3) receptors in living cells using a fluorescence-based binding assay.

Stoddart LA, Vernall AJ, Denman JL, Briddon SJ, Kellam B, Hill SJ. Stoddart LA, et al. Among authors: vernall aj. Chem Biol. 2012 Sep 21;19(9):1105-15. doi: 10.1016/j.chembiol.2012.07.014. Chem Biol. 2012. PMID: 22999879 Free PMC article.

4

The evolving small-molecule fluorescent-conjugate toolbox for Class A GPCRs.

Vernall AJ, Hill SJ, Kellam B. Vernall AJ, et al. Br J Pharmacol. 2014 Mar;171(5):1073-84. doi: 10.1111/bph.12265. Br J Pharmacol. 2014. PMID: 23734587 Free PMC article. Review.

5

Conversion of a non-selective adenosine receptor antagonist into A3-selective high affinity fluorescent probes using peptide-based linkers.

Vernall AJ, Stoddart LA, Briddon SJ, Ng HW, Laughton CA, Doughty SW, Hill SJ, Kellam B. Vernall AJ, et al. Org Biomol Chem. 2013 Sep 14;11(34):5673-82. doi: 10.1039/c3ob41221k. Org Biomol Chem. 2013. PMID: 23881285

6

Direct visualisation of internalization of the adenosine A3 receptor and localization with arrestin3 using a fluorescent agonist.

Stoddart LA, Vernall AJ, Briddon SJ, Kellam B, Hill SJ. Stoddart LA, et al. Among authors: vernall aj. Neuropharmacology. 2015 Nov;98:68-77. doi: 10.1016/j.neuropharm.2015.04.013. Epub 2015 Apr 30. Neuropharmacology. 2015. PMID: 25937210 Free article.

7

Chemical Tools for Studying Lipid-Binding Class A G Protein-Coupled Receptors.

Cooper A, Singh S, Hook S, Tyndall JDA, Vernall AJ. Cooper A, et al. Among authors: vernall aj. Pharmacol Rev. 2017 Jul;69(3):316-353. doi: 10.1124/pr.116.013243. Pharmacol Rev. 2017. PMID: 28655732 Review.

8

Development of novel fluorescent histamine H₁-receptor antagonists to study ligand-binding kinetics in living cells.

Stoddart LA, Vernall AJ, Bouzo-Lorenzo M, Bosma R, Kooistra AJ, de Graaf C, Vischer HF, Leurs R, Briddon SJ, Kellam B, Hill SJ. Stoddart LA, et al. Among authors: vernall aj. Sci Rep. 2018 Jan 25;8(1):1572. doi: 10.1038/s41598-018-19714-2. Sci Rep. 2018. PMID: 29371669 Free PMC article.

9

Alkyl indole-based cannabinoid type 2 receptor tools: Exploration of linker and fluorophore attachment.

Cooper AG, MacDonald C, Glass M, Hook S, Tyndall JDA, Vernall AJ. Cooper AG, et al. Among authors: vernall aj. Eur J Med Chem. 2018 Feb 10;145:770-789. doi: 10.1016/j.ejmech.2017.11.076. Epub 2017 Nov 28. Eur J Med Chem. 2018. PMID: 29407590

10

Development of selective, fluorescent cannabinoid type 2 receptor ligands based on a 1,8-naphthyridin-2-(1H)-one-3-carboxamide scaffold.

Cooper AG, Oyagawa CRM, Manning JJ, Singh S, Hook S, Grimsey NL, Glass M, Tyndall JDA, Vernall AJ. Cooper AG, et al. Among authors: vernall aj. Medchemcomm. 2018 Oct 23;9(12):2055-2067. doi: 10.1039/c8md00448j. eCollection 2018 Dec 1. Medchemcomm. 2018. PMID: 30647881 Free PMC article.

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