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Synthetic Peptides That Antagonize the Angiotensin-Converting Enzyme-2 (ACE-2) Interaction with SARS-CoV-2 Receptor Binding Spike Protein.
Sadremomtaz A, Al-Dahmani ZM, Ruiz-Moreno AJ, Monti A, Wang C, Azad T, Bell JC, Doti N, Velasco-Velázquez MA, de Jong D, de Jonge J, Smit J, Dömling A, van Goor H, Groves MR. Sadremomtaz A, et al. Among authors: domling a. J Med Chem. 2022 Feb 24;65(4):2836-2847. doi: 10.1021/acs.jmedchem.1c00477. Epub 2021 Jul 30. J Med Chem. 2022. PMID: 34328726 Free PMC article.
2,30-Bis(10H-indole) heterocycles: New p53/MDM2/MDMX antagonists.
Neochoritis CG, Wang K, Estrada-Ortiz N, Herdtweck E, Kubica K, Twarda A, Zak KM, Holak TA, Dömling A. Neochoritis CG, et al. Among authors: domling a. Bioorg Med Chem Lett. 2015 Dec 15;25(24):5661-6. doi: 10.1016/j.bmcl.2015.11.019. Bioorg Med Chem Lett. 2015. PMID: 26584879 Free PMC article.
Synthesis and Enantiomeric Separation of a Novel Spiroketal Derivative: A Potent Human Telomerase Inhibitor with High in Vitro Anticancer Activity.
Fuggetta MP, De Mico A, Cottarelli A, Morelli F, Zonfrillo M, Ulgheri F, Peluso P, Mannu A, Deligia F, Marchetti M, Roviello G, Reyes Romero A, Dömling A, Spanu P. Fuggetta MP, et al. Among authors: domling a. J Med Chem. 2016 Oct 13;59(19):9140-9149. doi: 10.1021/acs.jmedchem.6b01046. Epub 2016 Sep 19. J Med Chem. 2016. PMID: 27592503
The relevance of Ki calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor.
Wapenaar H, van den Bosch T, Leus NGJ, van der Wouden PE, Eleftheriadis N, Hermans J, Hailu GS, Rotili D, Mai A, Dömling A, Bischoff R, Haisma HJ, Dekker FJ. Wapenaar H, et al. Among authors: domling a. Eur J Med Chem. 2017 Aug 18;136:480-486. doi: 10.1016/j.ejmech.2017.05.015. Epub 2017 May 5. Eur J Med Chem. 2017. PMID: 28527406 Free PMC article.
Artificial Macrocycles as IL-17A/IL-17RA Antagonists.
Wang W, Groves MR, Dömling A. Wang W, et al. Among authors: domling a. Medchemcomm. 2018 Jan 1;9(1):22-26. doi: 10.1039/C7MD00464H. Epub 2017 Oct 25. Medchemcomm. 2018. PMID: 29750108 Free PMC article.
264 results