An aldol-based build/couple/pair strategy for the synthesis of medium- and large-sized rings: discovery of macrocyclic histone deacetylase inhibitors.
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Marcaurelle LA, et al. Among authors: haggarty sj.
J Am Chem Soc. 2010 Dec 1;132(47):16962-76. doi: 10.1021/ja105119r. Epub 2010 Nov 10.
J Am Chem Soc. 2010.
PMID: 21067169
Free PMC article.