Gmeiner P - Search Results

1

Bivalent ligands promote endosomal trafficking of the dopamine D3 receptor-neurotensin receptor 1 heterodimer.

Budzinski J, Maschauer S, Kobayashi H, Couvineau P, Vogt H, Gmeiner P, Roggenhofer A, Prante O, Bouvier M, Weikert D. Budzinski J, et al. Among authors: gmeiner p. Commun Biol. 2021 Sep 10;4(1):1062. doi: 10.1038/s42003-021-02574-4. Commun Biol. 2021. PMID: 34508168 Free PMC article.

2

Fused azaindole derivatives: molecular design, synthesis and in vitro pharmacology leading to the preferential dopamine D3 receptor agonist FAUC 725.

Löber S, Hübner H, Gmeiner P. Löber S, et al. Among authors: gmeiner p. Bioorg Med Chem Lett. 2002 Sep 2;12(17):2377-80. doi: 10.1016/s0960-894x(02)00390-6. Bioorg Med Chem Lett. 2002. PMID: 12161137

3

Interactive SAR studies: rational discovery of super-potent and highly selective dopamine D3 receptor antagonists and partial agonists.

Bettinetti L, Schlotter K, Hübner H, Gmeiner P. Bettinetti L, et al. Among authors: gmeiner p. J Med Chem. 2002 Oct 10;45(21):4594-7. doi: 10.1021/jm025558r. J Med Chem. 2002. PMID: 12361386

4

Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype.

Hocke C, Prante O, Löber S, Hübner H, Gmeiner P, Kuwert T. Hocke C, et al. Among authors: gmeiner p. Bioorg Med Chem Lett. 2004 Aug 2;14(15):3963-6. doi: 10.1016/j.bmcl.2004.05.052. Bioorg Med Chem Lett. 2004. PMID: 15225707

5

Parallel synthesis and biological screening of dopamine receptor ligands taking advantage of a click chemistry based BAL linker.

Bettinetti L, Löber S, Hübner H, Gmeiner P. Bettinetti L, et al. Among authors: gmeiner p. J Comb Chem. 2005 Mar-Apr;7(2):309-16. doi: 10.1021/cc049860s. J Comb Chem. 2005. PMID: 15762761

6

Fancy bioisosteres: synthesis, SAR, and pharmacological investigations of novel nonaromatic dopamine D3 receptor ligands.

Lenz C, Boeckler F, Hübner H, Gmeiner P. Lenz C, et al. Among authors: gmeiner p. Bioorg Med Chem. 2005 Jul 15;13(14):4434-42. doi: 10.1016/j.bmc.2005.04.047. Bioorg Med Chem. 2005. PMID: 15908220

7

Pharmacophore-guided drug discovery investigations leading to bioactive 5-aminotetrahydropyrazolopyridines. Implications for the binding mode of heterocyclic dopamine D3 receptor agonists.

Elsner J, Boeckler F, Heinemann FW, Hübner H, Gmeiner P. Elsner J, et al. Among authors: gmeiner p. J Med Chem. 2005 Sep 8;48(18):5771-9. doi: 10.1021/jm0503805. J Med Chem. 2005. PMID: 16134944

8

Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents.

Hocke C, Prante O, Löber S, Hübner H, Gmeiner P, Kuwert T. Hocke C, et al. Among authors: gmeiner p. Bioorg Med Chem Lett. 2005 Nov 1;15(21):4819-23. doi: 10.1016/j.bmcl.2005.07.037. Bioorg Med Chem Lett. 2005. PMID: 16139501

9

Tissue distribution of radioiodinated FAUC113: assessment of a pyrazolo(1,5-a) pyridine based dopamine D4 receptor radioligand candidate.

Prante O, Hocke C, Löber S, Hübner H, Gmeiner P, Kuwert T. Prante O, et al. Among authors: gmeiner p. Nuklearmedizin. 2006;45(1):41-8. doi: 10.1267/nukl06010041. Nuklearmedizin. 2006. PMID: 16493513

10

CoMFA and CoMSIA investigations of dopamine D3 receptor ligands leading to the prediction, synthesis, and evaluation of rigidized FAUC 365 analogues.

Salama I, Schlotter K, Utz W, Hübner H, Gmeiner P, Boeckler F. Salama I, et al. Among authors: gmeiner p. Bioorg Med Chem. 2006 Sep 1;14(17):5898-912. doi: 10.1016/j.bmc.2006.05.025. Epub 2006 Jun 5. Bioorg Med Chem. 2006. PMID: 16750374

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