Teleb M - Search Results

1

Halting Tumor Progression via Novel Non-Hydroxamate Triazole-Based Mannich Bases MMP-2/9 Inhibitors; Design, Microwave-Assisted Synthesis, and Biological Evaluation.

Albelwi FF, Teleb M, Abu-Serie MM, Moaty MNAA, Alsubaie MS, Zakaria MA, El Kilany Y, Aouad MR, Hagar M, Rezki N. Albelwi FF, et al. Among authors: teleb m. Int J Mol Sci. 2021 Sep 25;22(19):10324. doi: 10.3390/ijms221910324. Int J Mol Sci. 2021. PMID: 34638665 Free PMC article.

2

Chlorinated tacrine analogs: Design, synthesis and biological evaluation of their anti-cholinesterase activity as potential treatment for Alzheimer's disease.

Ragab HM, Teleb M, Haidar HR, Gouda N. Ragab HM, et al. Among authors: teleb m. Bioorg Chem. 2019 May;86:557-568. doi: 10.1016/j.bioorg.2019.02.033. Epub 2019 Feb 14. Bioorg Chem. 2019. PMID: 30782574

3

Design, synthesis and biological evaluation of novel α-acyloxy carboxamides via Passerini reaction as caspase 3/7 activators.

Salah Ayoup M, Wahby Y, Abdel-Hamid H, Ramadan ES, Teleb M, Abu-Serie MM, Noby A. Salah Ayoup M, et al. Among authors: teleb m. Eur J Med Chem. 2019 Apr 15;168:340-356. doi: 10.1016/j.ejmech.2019.02.051. Epub 2019 Feb 22. Eur J Med Chem. 2019. PMID: 30826510

4

Dual VEGFR-2/PIM-1 kinase inhibition towards surmounting the resistance to antiangiogenic agents via hybrid pyridine and thienopyridine-based scaffolds: Design, synthesis and biological evaluation.

Rizk OH, Teleb M, Abu-Serie MM, Shaaban OG. Rizk OH, et al. Among authors: teleb m. Bioorg Chem. 2019 Nov;92:103189. doi: 10.1016/j.bioorg.2019.103189. Epub 2019 Aug 8. Bioorg Chem. 2019. PMID: 31473473

5

Battle tactics against MMP-9; discovery of novel non-hydroxamate MMP-9 inhibitors endowed with PI3K/AKT signaling attenuation and caspase 3/7 activation via Ugi bis-amide synthesis.

Ayoup MS, Fouad MA, Abdel-Hamid H, Ramadan ES, Abu-Serie MM, Noby A, Teleb M. Ayoup MS, et al. Among authors: teleb m. Eur J Med Chem. 2020 Jan 15;186:111875. doi: 10.1016/j.ejmech.2019.111875. Epub 2019 Nov 10. Eur J Med Chem. 2020. PMID: 31740054

6

Structure-based design and optimization of pyrimidine- and 1,2,4-triazolo[4,3-a]pyrimidine-based matrix metalloproteinase-10/13 inhibitors via Dimroth rearrangement towards targeted polypharmacology.

El Ashry ESH, Awad LF, Teleb M, Ibrahim NA, Abu-Serie MM, Abd Al Moaty MN. El Ashry ESH, et al. Among authors: teleb m. Bioorg Chem. 2020 Mar;96:103616. doi: 10.1016/j.bioorg.2020.103616. Epub 2020 Jan 25. Bioorg Chem. 2020. PMID: 32032847

7

Beyond direct Nrf2 activation; reinvestigating 1,2,4-oxadiazole scaffold as a master key unlocking the antioxidant cellular machinery for cancer therapy.

Ayoup MS, Abu-Serie MM, Abdel-Hamid H, Teleb M. Ayoup MS, et al. Among authors: teleb m. Eur J Med Chem. 2021 Aug 5;220:113475. doi: 10.1016/j.ejmech.2021.113475. Epub 2021 Apr 16. Eur J Med Chem. 2021. PMID: 33901898

8

Halting colorectal cancer metastasis via novel dual nanomolar MMP-9/MAO-A quinoxaline-based inhibitors; design, synthesis, and evaluation.

Ayoup MS, Abu-Serie MM, Awad LF, Teleb M, Ragab HM, Amer A. Ayoup MS, et al. Among authors: teleb m. Eur J Med Chem. 2021 Oct 15;222:113558. doi: 10.1016/j.ejmech.2021.113558. Epub 2021 May 29. Eur J Med Chem. 2021. PMID: 34116327

9

Structural optimization, synthesis and in vitro synergistic anticancer activities of combinations of new N3-substituted dihydropyrimidine calcium channel blockers with cisplatin and etoposide.

El-Wakil MH, Teleb M, Abu-Serie MM, Huang S, Zamponi GW, Fahmy H. El-Wakil MH, et al. Among authors: teleb m. Bioorg Chem. 2021 Oct;115:105262. doi: 10.1016/j.bioorg.2021.105262. Epub 2021 Aug 11. Bioorg Chem. 2021. PMID: 34411980

10

Transforming Type II to Type I c-Met kinase inhibitors via combined scaffold hopping and structure-guided synthesis of new series of 1,3,4-thiadiazolo[2,3-c]-1,2,4-triazin-4-one derivatives.

El-Wakil MH, Teleb M. El-Wakil MH, et al. Among authors: teleb m. Bioorg Chem. 2021 Nov;116:105304. doi: 10.1016/j.bioorg.2021.105304. Epub 2021 Aug 25. Bioorg Chem. 2021. PMID: 34534756

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