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Development and Nanoparticle-Mediated Delivery of Novel MDM2/MDM4 Heterodimer Peptide Inhibitors to Enhance 5-Fluorouracil Nucleolar Stress in Colorectal Cancer Cells.
Merlino F, Pecoraro A, Longobardi G, Donati G, Di Leva FS, Brignola C, Piccarducci R, Daniele S, Martini C, Marinelli L, Russo G, Quaglia F, Conte C, Russo A, La Pietra V. Merlino F, et al. J Med Chem. 2024 Feb 8;67(3):1812-1824. doi: 10.1021/acs.jmedchem.3c01312. Epub 2024 Jan 29. J Med Chem. 2024. PMID: 38285632
From a Helix to a Small Cycle: Metadynamics-Inspired αvβ6 Integrin Selective Ligands.
Di Leva FS, Tomassi S, Di Maro S, Reichart F, Notni J, Dangi A, Marelli UK, Brancaccio D, Merlino F, Wester HJ, Novellino E, Kessler H, Marinelli L. Di Leva FS, et al. Among authors: merlino f. Angew Chem Int Ed Engl. 2018 Oct 26;57(44):14645-14649. doi: 10.1002/anie.201803250. Epub 2018 May 2. Angew Chem Int Ed Engl. 2018. PMID: 29660806
Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication.
Merlino F, Tomassi S, Yousif AM, Messere A, Marinelli L, Grieco P, Novellino E, Cosconati S, Di Maro S. Merlino F, et al. Org Lett. 2019 Aug 16;21(16):6378-6382. doi: 10.1021/acs.orglett.9b02283. Epub 2019 Jul 30. Org Lett. 2019. PMID: 31361506
Disulfide Bond Replacement with 1,4- and 1,5-Disubstituted [1,2,3]-Triazole on C-X-C Chemokine Receptor Type 4 (CXCR4) Peptide Ligands: Small Changes that Make Big Differences.
Tomassi S, Trotta AM, Ieranò C, Merlino F, Messere A, Rea G, Santoro F, Brancaccio D, Carotenuto A, D'Amore VM, Di Leva FS, Novellino E, Cosconati S, Marinelli L, Scala S, Di Maro S. Tomassi S, et al. Among authors: merlino f. Chemistry. 2020 Aug 6;26(44):10113-10125. doi: 10.1002/chem.202002468. Epub 2020 Jul 20. Chemistry. 2020. PMID: 32603023
Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides.
Merlino F, Billard É, Yousif AM, Di Maro S, Brancaccio D, Abate L, Carotenuto A, Bellavita R, d'Emmanuele di Villa Bianca R, Santicioli P, Marinelli L, Novellino E, Hébert TE, Lubell WD, Chatenet D, Grieco P. Merlino F, et al. J Med Chem. 2019 Feb 14;62(3):1455-1467. doi: 10.1021/acs.jmedchem.8b01601. Epub 2019 Jan 23. J Med Chem. 2019. PMID: 30615452
Simultaneous Targeting of RGD-Integrins and Dual Murine Double Minute Proteins in Glioblastoma Multiforme.
Merlino F, Daniele S, La Pietra V, Di Maro S, Di Leva FS, Brancaccio D, Tomassi S, Giuntini S, Cerofolini L, Fragai M, Luchinat C, Reichart F, Cavallini C, Costa B, Piccarducci R, Taliani S, Da Settimo F, Martini C, Kessler H, Novellino E, Marinelli L. Merlino F, et al. J Med Chem. 2018 Jun 14;61(11):4791-4809. doi: 10.1021/acs.jmedchem.8b00004. Epub 2018 Jun 4. J Med Chem. 2018. PMID: 29775303
Novel α-MSH peptide analogues with broad spectrum antimicrobial activity.
Grieco P, Carotenuto A, Auriemma L, Limatola A, Di Maro S, Merlino F, Mangoni ML, Luca V, Di Grazia A, Gatti S, Campiglia P, Gomez-Monterrey I, Novellino E, Catania A. Grieco P, et al. Among authors: merlino f. PLoS One. 2013 Apr 23;8(4):e61614. doi: 10.1371/journal.pone.0061614. Print 2013. PLoS One. 2013. PMID: 23626703 Free PMC article.
79 results