Gargano EM - Search Results

1

The 2-Methoxymethyl Modification of p -Phenylenediamine Reduces the Sensitization Risk for Hairdressers to Hair Dyes-An Occupational Hand Exposure-Based Risk Assessment.

Gargano EM, Blömeke B, Gaspari AA, Goebel C. Gargano EM, et al. Dermatitis. 2022 Jul-Aug 01;33(4):293-301. doi: 10.1097/DER.0000000000000915. Epub 2022 Jun 29. Dermatitis. 2022. PMID: 35777963 Free PMC article.

2

Development and validation of a method for simultaneous analysis of hair underivatized amino acids and damage biomarkers, using liquid chromatography-tandem mass spectrometry.

Gargano EM, Sell S, Langhoff S, Schmidt CU, Wierlacher S. Gargano EM, et al. Talanta. 2021 Oct 1;233:122584. doi: 10.1016/j.talanta.2021.122584. Epub 2021 Jun 8. Talanta. 2021. PMID: 34215076

3

Discovery of a Novel Potent and Selective HSD17B13 Inhibitor, BI-3231, a Well-Characterized Chemical Probe Available for Open Science.

Thamm S, Willwacher MK, Aspnes GE, Bretschneider T, Brown NF, Buschbom-Helmke S, Fox T, Gargano EM, Grabowski D, Hoenke C, Matera D, Mueck K, Peters S, Reindl S, Riether D, Schmid M, Tautermann CS, Teitelbaum AM, Trünkle C, Veser T, Winter M, Wortmann L. Thamm S, et al. Among authors: gargano em. J Med Chem. 2023 Feb 23;66(4):2832-2850. doi: 10.1021/acs.jmedchem.2c01884. Epub 2023 Feb 2. J Med Chem. 2023. PMID: 36727857 Free PMC article.

4

17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer.

Gargano EM, Mohamed A, Abdelsamie AS, Mangiatordi GF, Drzewiecka H, Jagodziński PP, Mazzini A, van Koppen CJ, Laschke MW, Nicolotti O, Carotti A, Marchais-Oberwinkler S, Hartmann RW, Frotscher M. Gargano EM, et al. ACS Med Chem Lett. 2021 Nov 18;12(12):1920-1924. doi: 10.1021/acsmedchemlett.1c00462. eCollection 2021 Dec 9. ACS Med Chem Lett. 2021. PMID: 34917255 Free PMC article.

5

Metabolism of the Selective Matrix Metalloproteinase-9 Inhibitor (R)-ND-336.

Gabriel CER, Nguyen TT, Gargano EM, Fisher JF, Chang M, Mobashery S. Gabriel CER, et al. Among authors: gargano em. ACS Pharmacol Transl Sci. 2021 Apr 6;4(3):1204-1213. doi: 10.1021/acsptsci.1c00063. eCollection 2021 Jun 11. ACS Pharmacol Transl Sci. 2021. PMID: 34151210 Free PMC article.

6

Persulfate Reaction in a Hair-Bleaching Formula: Unveiling the Unconventional Reactivity of 1,13-Diamino-4,7,10-Trioxatridecane.

Gargano EM, Mangiatordi GF, Weber I, Goebel C, Alberga D, Nicolotti O, Ruess W, Wierlacher S. Gargano EM, et al. ChemistryOpen. 2018 Mar 25;7(5):319-322. doi: 10.1002/open.201800013. eCollection 2018 May. ChemistryOpen. 2018. PMID: 29744283 Free PMC article.

7

Addressing cytotoxicity of 1,4-biphenyl amide derivatives: Discovery of new potent and selective 17β-hydroxysteroid dehydrogenase type 2 inhibitors.

Gargano EM, Perspicace E, Carotti A, Marchais-Oberwinkler S, Hartmann RW. Gargano EM, et al. Bioorg Med Chem Lett. 2016 Jan 1;26(1):21-4. doi: 10.1016/j.bmcl.2015.11.047. Epub 2015 Nov 23. Bioorg Med Chem Lett. 2016. PMID: 26615885

8

Towards the evaluation in an animal disease model: Fluorinated 17β-HSD1 inhibitors showing strong activity towards both the human and the rat enzyme.

Abdelsamie AS, Bey E, Gargano EM, van Koppen CJ, Empting M, Frotscher M. Abdelsamie AS, et al. Among authors: gargano em. Eur J Med Chem. 2015 Oct 20;103:56-68. doi: 10.1016/j.ejmech.2015.08.030. Epub 2015 Aug 18. Eur J Med Chem. 2015. PMID: 26322835

9

17β-Hydroxysteroid Dehydrogenase Type 2 Inhibition: Discovery of Selective and Metabolically Stable Compounds Inhibiting Both the Human Enzyme and Its Murine Ortholog.

Gargano EM, Allegretta G, Perspicace E, Carotti A, Van Koppen C, Frotscher M, Marchais-Oberwinkler S, Hartmann RW. Gargano EM, et al. PLoS One. 2015 Jul 31;10(7):e0134754. doi: 10.1371/journal.pone.0134754. eCollection 2015. PLoS One. 2015. PMID: 26230928 Free PMC article.

10

Metabolic stability optimization and metabolite identification of 2,5-thiophene amide 17β-hydroxysteroid dehydrogenase type 2 inhibitors.

Gargano EM, Perspicace E, Hanke N, Carotti A, Marchais-Oberwinkler S, Hartmann RW. Gargano EM, et al. Eur J Med Chem. 2014 Nov 24;87:203-19. doi: 10.1016/j.ejmech.2014.09.061. Epub 2014 Sep 20. Eur J Med Chem. 2014. PMID: 25259513

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