Daelemans D - Search Results

1

Imidazo[4,5-b]pyridine derived tubulin polymerization inhibitors: Design, synthesis, biological activity in vitro and computational analysis.

Boček I, Hok L, Persoons L, Daelemans D, Vianello R, Hranjec M. Boček I, et al. Among authors: daelemans d. Bioorg Chem. 2022 Oct;127:106032. doi: 10.1016/j.bioorg.2022.106032. Epub 2022 Jul 16. Bioorg Chem. 2022. PMID: 35872398

2

Allosteric degraders induce CRL5 ^ASB8 mediated degradation of XPO1.

Hudman-Wing CE, Fung HYJ, Cagatay T, Kwanten B, Niesman AB, Gharghabi M, Permentier B, Shakya B, Shacham S, Landesman Y, Lapalombella R, Daelemans D, Chook YM. Hudman-Wing CE, et al. Among authors: daelemans d. bioRxiv [Preprint]. 2024 Oct 11:2024.10.07.617049. doi: 10.1101/2024.10.07.617049. bioRxiv. 2024. PMID: 39416201 Free PMC article. Preprint.

3

Inhibition of the CRM1-mediated nucleocytoplasmic transport by N-azolylacrylates: structure-activity relationship and mechanism of action.

Van Neck T, Pannecouque C, Vanstreels E, Stevens M, Dehaen W, Daelemans D. Van Neck T, et al. Among authors: daelemans d. Bioorg Med Chem. 2008 Nov 1;16(21):9487-97. doi: 10.1016/j.bmc.2008.09.051. Epub 2008 Sep 20. Bioorg Med Chem. 2008. PMID: 18835718

4

Towards new C6-rigid S-DABO HIV-1 reverse transcriptase inhibitors: synthesis, biological investigation and molecular modeling studies.

Wu HQ, Yan ZH, Chen WX, He QQ, Chen FE, De Clercq E, Balzarini J, Daelemans D, Pannecouque C. Wu HQ, et al. Among authors: daelemans d. Bioorg Med Chem. 2013 Nov 1;21(21):6477-83. doi: 10.1016/j.bmc.2013.08.040. Epub 2013 Aug 30. Bioorg Med Chem. 2013. PMID: 24055077

5

Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands.

Sancineto L, Iraci N, Barreca ML, Massari S, Manfroni G, Corazza G, Cecchetti V, Marcello A, Daelemans D, Pannecouque C, Tabarrini O. Sancineto L, et al. Among authors: daelemans d. Bioorg Med Chem. 2014 Sep 1;22(17):4658-66. doi: 10.1016/j.bmc.2014.07.018. Epub 2014 Jul 22. Bioorg Med Chem. 2014. PMID: 25127466

6

Synthesis and biological evaluation of DAPY-DPEs hybrids as non-nucleoside inhibitors of HIV-1 reverse transcriptase.

Wu HQ, Yao J, He QQ, Chen WX, Chen FE, Pannecouque C, De Clercq E, Daelemans D. Wu HQ, et al. Among authors: daelemans d. Bioorg Med Chem. 2015 Feb 1;23(3):624-31. doi: 10.1016/j.bmc.2014.11.032. Epub 2014 Nov 27. Bioorg Med Chem. 2015. PMID: 25537532

7

Hybrid chemistry. Part 4: Discovery of etravirine-VRX-480773 hybrids as potent HIV-1 non-nucleoside reverse transcriptase inhibitors.

Wan ZY, Tao Y, Wang YF, Mao TQ, Yin H, Chen FE, Piao HR, De Clercq E, Daelemans D, Pannecouque C. Wan ZY, et al. Among authors: daelemans d. Bioorg Med Chem. 2015 Aug 1;23(15):4248-4255. doi: 10.1016/j.bmc.2015.06.048. Epub 2015 Jun 27. Bioorg Med Chem. 2015. PMID: 26162497

8

L-Aspartic and l-glutamic acid ester-based ProTides of anticancer nucleosides: Synthesis and antitumoral evaluation.

Gao LJ, De Jonghe S, Daelemans D, Herdewijn P. Gao LJ, et al. Among authors: daelemans d. Bioorg Med Chem Lett. 2016 May 1;26(9):2142-6. doi: 10.1016/j.bmcl.2016.03.076. Epub 2016 Mar 22. Bioorg Med Chem Lett. 2016. PMID: 27032331

9

Arylazolyl(azinyl)thioacetanilides. Part 20: Discovery of novel purinylthioacetanilides derivatives as potent HIV-1 NNRTIs via a structure-based bioisosterism approach.

Lu X, Li X, Yang J, Huang B, Kang D, Zhao F, Zhou Z, De Clercq E, Daelemans D, Pannecouque C, Zhan P, Liu X. Lu X, et al. Among authors: daelemans d. Bioorg Med Chem. 2016 Sep 15;24(18):4424-4433. doi: 10.1016/j.bmc.2016.07.041. Epub 2016 Jul 21. Bioorg Med Chem. 2016. PMID: 27501911

10

Discovery of novel DAPY-IAS hybrid derivatives as potential HIV-1 inhibitors using molecular hybridization based on crystallographic overlays.

Huang B, Wang X, Liu X, Chen Z, Li W, Sun S, Liu H, Daelemans D, De Clercq E, Pannecouque C, Zhan P, Liu X. Huang B, et al. Among authors: daelemans d. Bioorg Med Chem. 2017 Aug 15;25(16):4397-4406. doi: 10.1016/j.bmc.2017.06.022. Epub 2017 Jun 15. Bioorg Med Chem. 2017. PMID: 28659246

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