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Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment.
Di Maria S, Picarazzi F, Mori M, Cianciusi A, Carbone A, Crespan E, Perini C, Sabetta S, Deplano S, Poggialini F, Molinari A, Aronne R, Maccioni E, Maga G, Angelucci A, Schenone S, Musumeci F, Dreassi E. Di Maria S, et al. Among authors: deplano s. Bioorg Chem. 2022 Nov;128:106071. doi: 10.1016/j.bioorg.2022.106071. Epub 2022 Aug 1. Bioorg Chem. 2022. PMID: 35932498
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation.
Fois B, Distinto S, Meleddu R, Deplano S, Maccioni E, Floris C, Rosa A, Nieddu M, Caboni P, Sissi C, Angeli A, Supuran CT, Cottiglia F. Fois B, et al. Among authors: deplano s. J Enzyme Inhib Med Chem. 2020 Dec;35(1):539-548. doi: 10.1080/14756366.2020.1713114. J Enzyme Inhib Med Chem. 2020. PMID: 31948300 Free PMC article.
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives.
Meleddu R, Deplano S, Maccioni E, Ortuso F, Cottiglia F, Secci D, Onali A, Sanna E, Angeli A, Angius R, Alcaro S, Supuran CT, Distinto S. Meleddu R, et al. Among authors: deplano s. J Enzyme Inhib Med Chem. 2021 Dec;36(1):685-692. doi: 10.1080/14756366.2021.1887171. J Enzyme Inhib Med Chem. 2021. PMID: 33602041 Free PMC article.
New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII.
Meleddu R, Distinto S, Cottiglia F, Angius R, Caboni P, Angeli A, Melis C, Deplano S, Alcaro S, Ortuso F, Supuran CT, Maccioni E. Meleddu R, et al. Among authors: deplano s. ACS Med Chem Lett. 2020 Feb 13;11(5):852-856. doi: 10.1021/acsmedchemlett.9b00644. eCollection 2020 May 14. ACS Med Chem Lett. 2020. PMID: 32435395 Free PMC article.
Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids.
Meleddu R, Petrikaite V, Distinto S, Arridu A, Angius R, Serusi L, Škarnulytė L, Endriulaitytė U, Paškevičiu Tė M, Cottiglia F, Gaspari M, Taverna D, Deplano S, Fois B, Maccioni E. Meleddu R, et al. Among authors: deplano s. ACS Med Chem Lett. 2018 Dec 18;10(4):571-576. doi: 10.1021/acsmedchemlett.8b00596. eCollection 2019 Apr 11. ACS Med Chem Lett. 2018. PMID: 30996798 Free PMC article.
Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides.
Meleddu R, Distinto S, Cottiglia F, Angius R, Gaspari M, Taverna D, Melis C, Angeli A, Bianco G, Deplano S, Fois B, Del Prete S, Capasso C, Alcaro S, Ortuso F, Yanez M, Supuran CT, Maccioni E. Meleddu R, et al. Among authors: deplano s. ACS Med Chem Lett. 2018 Sep 17;9(10):1045-1050. doi: 10.1021/acsmedchemlett.8b00352. eCollection 2018 Oct 11. ACS Med Chem Lett. 2018. PMID: 30344915 Free PMC article.
Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases.
Distinto S, Meleddu R, Ortuso F, Cottiglia F, Deplano S, Sequeira L, Melis C, Fois B, Angeli A, Capasso C, Angius R, Alcaro S, Supuran CT, Maccioni E. Distinto S, et al. Among authors: deplano s. J Enzyme Inhib Med Chem. 2019 Dec;34(1):1526-1533. doi: 10.1080/14756366.2019.1654470. J Enzyme Inhib Med Chem. 2019. PMID: 31431095 Free PMC article.
45 results