Colarusso E - Search Results

1

Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders.

Colarusso E, Ceccacci S, Monti MC, Gazzillo E, Giordano A, Chini MG, Ferraro MG, Piccolo M, Ruggiero D, Irace C, Terracciano S, Bruno I, Bifulco G, Lauro G. Colarusso E, et al. Eur J Med Chem. 2023 Feb 5;247:115018. doi: 10.1016/j.ejmech.2022.115018. Epub 2022 Dec 17. Eur J Med Chem. 2023. PMID: 36577218

2

Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE₂ Levels.

Chini MG, Giordano A, Potenza M, Terracciano S, Fischer K, Vaccaro MC, Colarusso E, Bruno I, Riccio R, Koeberle A, Werz O, Bifulco G. Chini MG, et al. Among authors: colarusso e. ACS Med Chem Lett. 2020 Mar 5;11(5):783-789. doi: 10.1021/acsmedchemlett.9b00618. eCollection 2020 May 14. ACS Med Chem Lett. 2020. PMID: 32435385 Free PMC article.

3

Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9.

Gazzillo E, Pierri M, Colarusso E, Chini MG, Ferraro MG, Piccolo M, Irace C, Bruno I, Bifulco G, Terracciano S, Lauro G. Gazzillo E, et al. Among authors: colarusso e. Bioorg Chem. 2023 Oct;139:106677. doi: 10.1016/j.bioorg.2023.106677. Epub 2023 Jun 12. Bioorg Chem. 2023. PMID: 37352721 Free article.

4

2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines.

De Vita S, Meninno S, Capasso L, Colarusso E, Chini MG, Lauro G, Rinaldi R, De Cicco A, Sian V, Terracciano S, Nebbioso A, Lattanzi A, Bifulco G. De Vita S, et al. Among authors: colarusso e. Bioorg Med Chem. 2023 Oct 1;93:117444. doi: 10.1016/j.bmc.2023.117444. Epub 2023 Aug 12. Bioorg Med Chem. 2023. PMID: 37611334 Free article.

5

Identification and Development of BRD9 Chemical Probes.

Colarusso E, Chini MG, Bifulco G, Lauro G, Giordano A. Colarusso E, et al. Pharmaceuticals (Basel). 2024 Mar 19;17(3):392. doi: 10.3390/ph17030392. Pharmaceuticals (Basel). 2024. PMID: 38543178 Free PMC article. Review.

6

PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes.

De Vita S, Colarusso E, Chini MG, Bifulco G, Lauro G. De Vita S, et al. Among authors: colarusso e. J Chem Inf Model. 2024 May 27;64(10):4263-4276. doi: 10.1021/acs.jcim.3c01920. Epub 2024 May 10. J Chem Inf Model. 2024. PMID: 38728062

7

Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH).

Gazzillo E, Colarusso E, Giordano A, Chini MG, Potenza M, Hofstetter RK, Iorizzi M, Werz O, Lauro G, Bifulco G. Gazzillo E, et al. Among authors: colarusso e. Chempluschem. 2024 Sep;89(9):e202400234. doi: 10.1002/cplu.202400234. Epub 2024 Jun 11. Chempluschem. 2024. PMID: 38753468

8

Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition.

Fantasma F, Samukha V, Aliberti M, Colarusso E, Chini MG, Saviano G, De Felice V, Lauro G, Casapullo A, Bifulco G, Iorizzi M. Fantasma F, et al. Among authors: colarusso e. Foods. 2024 Jul 20;13(14):2282. doi: 10.3390/foods13142282. Foods. 2024. PMID: 39063366 Free PMC article.

9

In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders.

Colarusso E, Gazzillo E, Pierri M, Ruggiero D, Chini MG, Bruno I, Bifulco G, Terracciano S, Lauro G. Colarusso E, et al. Chempluschem. 2024 Dec;89(12):e202400339. doi: 10.1002/cplu.202400339. Epub 2024 Oct 18. Chempluschem. 2024. PMID: 39119716

10

Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign.

Colarusso E, Gazzillo E, Boccia E, Terracciano S, Bruno I, Bifulco G, Chini MG, Lauro G. Colarusso E, et al. Molecules. 2024 Aug 26;29(17):4025. doi: 10.3390/molecules29174025. Molecules. 2024. PMID: 39274873 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

18 results

Search Page

Filters