Lauro G - Search Results

1

Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders.

Colarusso E, Ceccacci S, Monti MC, Gazzillo E, Giordano A, Chini MG, Ferraro MG, Piccolo M, Ruggiero D, Irace C, Terracciano S, Bruno I, Bifulco G, Lauro G. Colarusso E, et al. Among authors: lauro g. Eur J Med Chem. 2023 Feb 5;247:115018. doi: 10.1016/j.ejmech.2022.115018. Epub 2022 Dec 17. Eur J Med Chem. 2023. PMID: 36577218

2

Inverse virtual screening of antitumor targets: pilot study on a small database of natural bioactive compounds.

Lauro G, Romano A, Riccio R, Bifulco G. Lauro G, et al. J Nat Prod. 2011 Jun 24;74(6):1401-7. doi: 10.1021/np100935s. Epub 2011 May 4. J Nat Prod. 2011. PMID: 21542600

3

Discovery and synthesis of namalide reveals a new anabaenopeptin scaffold and peptidase inhibitor.

Cheruku P, Plaza A, Lauro G, Keffer J, Lloyd JR, Bifulco G, Bewley CA. Cheruku P, et al. Among authors: lauro g. J Med Chem. 2012 Jan 26;55(2):735-42. doi: 10.1021/jm201238p. Epub 2012 Jan 5. J Med Chem. 2012. PMID: 22168797 Free PMC article.

4

Inverse Virtual Screening allows the discovery of the biological activity of natural compounds.

Lauro G, Masullo M, Piacente S, Riccio R, Bifulco G. Lauro G, et al. Bioorg Med Chem. 2012 Jun 1;20(11):3596-602. doi: 10.1016/j.bmc.2012.03.072. Epub 2012 Apr 6. Bioorg Med Chem. 2012. PMID: 22537682

5

Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist.

Sepe V, Ummarino R, D'Auria MV, Lauro G, Bifulco G, D'Amore C, Renga B, Fiorucci S, Zampella A. Sepe V, et al. Among authors: lauro g. Org Biomol Chem. 2012 Aug 21;10(31):6350-62. doi: 10.1039/c2ob25800e. Epub 2012 Jun 26. Org Biomol Chem. 2012. PMID: 22733410

6

Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ.

Festa C, Lauro G, De Marino S, D'Auria MV, Monti MC, Casapullo A, D'Amore C, Renga B, Mencarelli A, Petek S, Bifulco G, Fiorucci S, Zampella A. Festa C, et al. Among authors: lauro g. J Med Chem. 2012 Oct 11;55(19):8303-17. doi: 10.1021/jm300911g. Epub 2012 Sep 19. J Med Chem. 2012. PMID: 22934537

7

Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells.

Dal Piaz F, Cotugno R, Lepore L, Vassallo A, Malafronte N, Lauro G, Bifulco G, Belisario MA, De Tommasi N. Dal Piaz F, et al. Among authors: lauro g. J Proteomics. 2013 Apr 26;82:14-26. doi: 10.1016/j.jprot.2013.01.030. Epub 2013 Feb 15. J Proteomics. 2013. PMID: 23416714

8

Oxygenated polyketides from Plakinastrella mamillaris as a new chemotype of PXR agonists.

Festa C, D'Amore C, Renga B, Lauro G, De Marino S, D'Auria MV, Bifulco G, Zampella A, Fiorucci S. Festa C, et al. Among authors: lauro g. Mar Drugs. 2013 Jul 2;11(7):2314-27. doi: 10.3390/md11072314. Mar Drugs. 2013. PMID: 23820629 Free PMC article.

9

Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E₂ synthase-1 enzyme (mPGES-1).

Lauro G, Strocchia M, Terracciano S, Bruno I, Fischer K, Pergola C, Werz O, Riccio R, Bifulco G. Lauro G, et al. Eur J Med Chem. 2014 Jun 10;80:407-15. doi: 10.1016/j.ejmech.2014.04.061. Epub 2014 Apr 24. Eur J Med Chem. 2014. PMID: 24794772

10

Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A₂, cyclooxygenases, lipoxygenase and proinflammatory cytokines.

Bukhari SN, Lauro G, Jantan I, Bifulco G, Amjad MW. Bukhari SN, et al. Among authors: lauro g. Bioorg Med Chem. 2014 Aug 1;22(15):4151-61. doi: 10.1016/j.bmc.2014.05.052. Epub 2014 Jun 2. Bioorg Med Chem. 2014. PMID: 24938495

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