Cai M - Search Results

1

Ψ and χ Angle Constrains at the C-Terminus Trp Position of the Melanotropin Tetrapeptide Ac-His-d-Phe-Arg-Trp-NH₂ Lead to Potent and Selective Agonists at hMC1R and hMC4R.

Zhou Y, Mowlazadeh Haghighi S, Sawyer JR, Hruby VJ, Cai M. Zhou Y, et al. Among authors: cai m. J Med Chem. 2023 May 25;66(10):6715-6724. doi: 10.1021/acs.jmedchem.2c01794. Epub 2023 May 3. J Med Chem. 2023. PMID: 37133411

2

Novel cyclic templates of alpha-MSH give highly selective and potent antagonists/agonists for human melanocortin-3/4 receptors.

Kavarana MJ, Trivedi D, Cai M, Ying J, Hammer M, Cabello C, Grieco P, Han G, Hruby VJ. Kavarana MJ, et al. Among authors: cai m. J Med Chem. 2002 Jun 6;45(12):2644-50. doi: 10.1021/jm020021z. J Med Chem. 2002. PMID: 12036373

3

Structure-activity studies of the melanocortin peptides: discovery of potent and selective affinity antagonists for the hMC3 and hMC4 receptors.

Grieco P, Lavecchia A, Cai M, Trivedi D, Weinberg D, MacNeil T, Van der Ploeg LH, Hruby VJ. Grieco P, et al. Among authors: cai m. J Med Chem. 2002 Nov 21;45(24):5287-94. doi: 10.1021/jm0202526. J Med Chem. 2002. PMID: 12431055

4

Exploring the stereostructural requirements of peptide ligands for the melanocortin receptors.

Hruby VJ, Cai M, Grieco P, Han G, Kavarana M, Trivedi D. Hruby VJ, et al. Among authors: cai m. Ann N Y Acad Sci. 2003 Jun;994:12-20. doi: 10.1111/j.1749-6632.2003.tb03157.x. Ann N Y Acad Sci. 2003. PMID: 12851293

5

Structure-activity relationships of novel cyclic alpha-MSH/beta-MSH hybrid analogues that lead to potent and selective ligands for the human MC3R and human MC5R.

Balse-Srinivasan P, Grieco P, Cai M, Trivedi D, Hruby VJ. Balse-Srinivasan P, et al. Among authors: cai m. J Med Chem. 2003 Aug 14;46(17):3728-33. doi: 10.1021/jm030111j. J Med Chem. 2003. PMID: 12904077

6

Structure-activity relationships of gamma-MSH analogues at the human melanocortin MC3, MC4, and MC5 receptors. Discovery of highly selective hMC3R, hMC4R, and hMC5R analogues.

Balse-Srinivasan P, Grieco P, Cai M, Trivedi D, Hruby VJ. Balse-Srinivasan P, et al. Among authors: cai m. J Med Chem. 2003 Nov 6;46(23):4965-73. doi: 10.1021/jm030119t. J Med Chem. 2003. PMID: 14584947

7

Biological and conformational study of beta-substituted prolines in MT-II template: steric effects leading to human MC5 receptor selectivity.

Cai M, Cai C, Mayorov AV, Xiong C, Cabello CM, Soloshonok VA, Swift JR, Trivedi D, Hruby VJ. Cai M, et al. Among authors: cai c. J Pept Res. 2004 Feb;63(2):116-31. doi: 10.1111/j.1399-3011.2003.00105.x. J Pept Res. 2004. PMID: 15009533

8

Real time differentiation of G-protein coupled receptor (GPCR) agonist and antagonist by two photon fluorescence laser microscopy.

Cai M, Stankova M, Pond SJ, Mayorov AV, Perry JW, Yamamura HI, Trivedi D, Hruby VJ. Cai M, et al. J Am Chem Soc. 2004 Jun 16;126(23):7160-1. doi: 10.1021/ja049473m. J Am Chem Soc. 2004. PMID: 15186137

9

Novel 3D pharmacophore of alpha-MSH/gamma-MSH hybrids leads to selective human MC1R and MC3R analogues.

Cai M, Mayorov AV, Cabello C, Stankova M, Trivedi D, Hruby VJ. Cai M, et al. J Med Chem. 2005 Mar 24;48(6):1839-48. doi: 10.1021/jm049579s. J Med Chem. 2005. PMID: 15771429

10

Design of novel melanotropin agonists and antagonists with high potency and selectivity for human melanocortin receptors.

Cai M, Mayorov AV, Ying J, Stankova M, Trivedi D, Cabello C, Hruby VJ. Cai M, et al. Peptides. 2005 Aug;26(8):1481-5. doi: 10.1016/j.peptides.2005.03.020. Peptides. 2005. PMID: 15876475 Review.

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