Jacobson KA - Search Results

1

Assay-Dependent Inverse Agonism at the A₃ Adenosine Receptor: When Neutral Is Not Neutral.

Pottie E, Suresh RR, Jacobson KA, Stove CP. Pottie E, et al. Among authors: jacobson ka. ACS Pharmacol Transl Sci. 2023 Aug 9;6(9):1266-1274. doi: 10.1021/acsptsci.3c00071. eCollection 2023 Sep 8. ACS Pharmacol Transl Sci. 2023. PMID: 37705594 Free PMC article.

2

Flexible modulation of agonist efficacy at the human A3 adenosine receptor by the imidazoquinoline allosteric enhancer LUF6000.

Gao ZG, Ye K, Göblyös A, Ijzerman AP, Jacobson KA. Gao ZG, et al. Among authors: jacobson ka. BMC Pharmacol. 2008 Dec 12;8:20. doi: 10.1186/1471-2210-8-20. BMC Pharmacol. 2008. PMID: 19077268 Free PMC article.

3

Identification of A3 adenosine receptor agonists as novel non-narcotic analgesics.

Janes K, Symons-Liguori AM, Jacobson KA, Salvemini D. Janes K, et al. Among authors: jacobson ka. Br J Pharmacol. 2016 Apr;173(8):1253-67. doi: 10.1111/bph.13446. Epub 2016 Mar 6. Br J Pharmacol. 2016. PMID: 26804983 Free PMC article. Review.

4

Structure-Activity Analysis of Biased Agonism at the Human Adenosine A3 Receptor.

Baltos JA, Paoletta S, Nguyen AT, Gregory KJ, Tosh DK, Christopoulos A, Jacobson KA, May LT. Baltos JA, et al. Among authors: jacobson ka. Mol Pharmacol. 2016 Jul;90(1):12-22. doi: 10.1124/mol.116.103283. Epub 2016 May 2. Mol Pharmacol. 2016. PMID: 27136943 Free PMC article.

5

A binding kinetics study of human adenosine A₃ receptor agonists.

Xia L, Kyrizaki A, Tosh DK, van Duijl TT, Roorda JC, Jacobson KA, IJzerman AP, Heitman LH. Xia L, et al. Among authors: jacobson ka. Biochem Pharmacol. 2018 Jul;153:248-259. doi: 10.1016/j.bcp.2017.12.026. Epub 2018 Jan 3. Biochem Pharmacol. 2018. PMID: 29305857 Free PMC article.

6

Activation of adenosine A_2A or A_2B receptors causes hypothermia in mice.

Carlin JL, Jain S, Duroux R, Suresh RR, Xiao C, Auchampach JA, Jacobson KA, Gavrilova O, Reitman ML. Carlin JL, et al. Among authors: jacobson ka. Neuropharmacology. 2018 Sep 1;139:268-278. doi: 10.1016/j.neuropharm.2018.02.035. Epub 2018 Mar 13. Neuropharmacology. 2018. PMID: 29548686 Free PMC article.

7

Probing structure-activity relationship in β-arrestin2 recruitment of diversely substituted adenosine derivatives.

Storme J, Tosh DK, Gao ZG, Jacobson KA, Stove CP. Storme J, et al. Among authors: jacobson ka. Biochem Pharmacol. 2018 Dec;158:103-113. doi: 10.1016/j.bcp.2018.10.003. Epub 2018 Oct 4. Biochem Pharmacol. 2018. PMID: 30292756 Free PMC article.

8

Evidence for the Interaction of A₃ Adenosine Receptor Agonists at the Drug-Binding Site(s) of Human P-glycoprotein (ABCB1).

Abel B, Tosh DK, Durell SR, Murakami M, Vahedi S, Jacobson KA, Ambudkar SV. Abel B, et al. Among authors: jacobson ka. Mol Pharmacol. 2019 Aug;96(2):180-192. doi: 10.1124/mol.118.115295. Epub 2019 May 24. Mol Pharmacol. 2019. PMID: 31127007 Free PMC article.

9

Assessment of biased agonism at the A₃ adenosine receptor using β-arrestin and miniGα_i recruitment assays.

Pottie E, Tosh DK, Gao ZG, Jacobson KA, Stove CP. Pottie E, et al. Among authors: jacobson ka. Biochem Pharmacol. 2020 Jul;177:113934. doi: 10.1016/j.bcp.2020.113934. Epub 2020 Mar 26. Biochem Pharmacol. 2020. PMID: 32224136 Free PMC article.

10

Allosteric Antagonism of the A_2A Adenosine Receptor by a Series of Bitopic Ligands.

Gao ZG, Toti KS, Campbell R, Suresh RR, Yang H, Jacobson KA. Gao ZG, et al. Among authors: jacobson ka. Cells. 2020 May 12;9(5):1200. doi: 10.3390/cells9051200. Cells. 2020. PMID: 32408534 Free PMC article.

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