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Page 1
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors.
Di Stefano M, Masoni S, Bononi G, Poli G, Galati S, Gado F, Manzi S, Vagaggini C, Brai A, Caligiuri I, Asif K, Rizzolio F, Macchia M, Chicca A, Sodi A, Di Bussolo V, Minutolo F, Meier P, Gertsch J, Granchi C, Dreassi E, Tuccinardi T. Di Stefano M, et al. Among authors: dreassi e. Eur J Med Chem. 2024 Jan 5;263:115916. doi: 10.1016/j.ejmech.2023.115916. Epub 2023 Nov 2. Eur J Med Chem. 2024. PMID: 37976705 Free article.
Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma.
Di Maria S, Passannanti R, Poggialini F, Vagaggini C, Serafinelli A, Bianchi E, Governa P, Botta L, Maga G, Crespan E, Manetti F, Dreassi E, Musumeci F, Carbone A, Schenone S. Di Maria S, et al. Among authors: dreassi e. Eur J Med Chem. 2024 Dec 15;280:116929. doi: 10.1016/j.ejmech.2024.116929. Epub 2024 Oct 1. Eur J Med Chem. 2024. PMID: 39406114 Free article.
Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study.
Marinacci B, D'Agostino I, Angeli A, Carradori S, Melfi F, Grande R, Corsiani M, Ferraroni M, Agamennone M, Tondo AR, Zara S, Puca V, Pellegrini B, Vagaggini C, Dreassi E, Patrauchan MA, Capasso C, Nicolotti O, Carta F, Supuran CT. Marinacci B, et al. Among authors: dreassi e. J Med Chem. 2024 Nov 14;67(21):19077-19102. doi: 10.1021/acs.jmedchem.4c01555. Epub 2024 Oct 25. J Med Chem. 2024. PMID: 39453626
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth.
Maresca L, Crivaro E, Migliorini F, Anichini G, Giammona A, Pepe S, Poggialini F, Vagaggini C, Giannini G, Sestini S, Borgognoni L, Lapucci A, Dreassi E, Taddei M, Manetti F, Petricci E, Stecca B. Maresca L, et al. Among authors: dreassi e. Pharmacol Res. 2023 Sep;195:106858. doi: 10.1016/j.phrs.2023.106858. Epub 2023 Jul 19. Pharmacol Res. 2023. PMID: 37473878 Free article.
Optimization of potent, broad-spectrum, and specific anti-influenza compounds targeting RNA polymerase PA-PB1 heterodimerization.
Bonomini A, Felicetti T, Pacetti M, Bertagnin C, Coletti A, Giammarino F, De Angelis M, Poggialini F, Macchiarulo A, Sabatini S, Mercorelli B, Nencioni L, Vicenti I, Dreassi E, Cecchetti V, Tabarrini O, Loregian A, Massari S. Bonomini A, et al. Among authors: dreassi e. Eur J Med Chem. 2024 Nov 5;277:116737. doi: 10.1016/j.ejmech.2024.116737. Epub 2024 Aug 3. Eur J Med Chem. 2024. PMID: 39153334
127 results