Burke AJ - Search Results

1

Early pharmacological profiling of isatin derivatives as potent and selective cytotoxic agents.

Puerta A, González-Bakker A, Brandão P, Pineiro M, Burke AJ, Giovannetti E, Fernandes MX, Padrón JM. Puerta A, et al. Among authors: burke aj. Biochem Pharmacol. 2024 Apr;222:116059. doi: 10.1016/j.bcp.2024.116059. Epub 2024 Feb 15. Biochem Pharmacol. 2024. PMID: 38364984 Free article.

2

The application of isatin-based multicomponent-reactions in the quest for new bioactive and druglike molecules.

Brandão P, Marques C, Burke AJ, Pineiro M. Brandão P, et al. Among authors: burke aj. Eur J Med Chem. 2021 Feb 5;211:113102. doi: 10.1016/j.ejmech.2020.113102. Epub 2020 Dec 18. Eur J Med Chem. 2021. PMID: 33421712 Review.

3

Engaging Isatins in Multicomponent Reactions (MCRs) - Easy Access to Structural Diversity.

Brandão P, Marques CS, Carreiro EP, Pineiro M, Burke AJ. Brandão P, et al. Among authors: burke aj. Chem Rec. 2021 Apr;21(4):924-1037. doi: 10.1002/tcr.202000167. Epub 2021 Feb 18. Chem Rec. 2021. PMID: 33599390

4

Ugi Reaction Synthesis of Oxindole-Lactam Hybrids as Selective Butyrylcholinesterase Inhibitors.

Brandão P, López Ó, Leitzbach L, Stark H, Fernández-Bolaños JG, Burke AJ, Pineiro M. Brandão P, et al. Among authors: burke aj. ACS Med Chem Lett. 2021 Jul 23;12(11):1718-1725. doi: 10.1021/acsmedchemlett.1c00344. eCollection 2021 Nov 11. ACS Med Chem Lett. 2021. PMID: 34795859 Free PMC article.

5

Targeting Vascular Endothelial Growth Factor Receptor 2 (VEGFR-2): Latest Insights on Synthetic Strategies.

Marques CS, Brandão P, Burke AJ. Marques CS, et al. Among authors: burke aj. Molecules. 2024 Nov 13;29(22):5341. doi: 10.3390/molecules29225341. Molecules. 2024. PMID: 39598729 Free PMC article. Review.

6

N-1,2,3-Triazole-isatin derivatives: anti-proliferation effects and target identification in solid tumour cell lines.

Busto N, Leitão-Castro J, García-Sosa AT, Cadete F, Marques CS, Freitas R, Burke AJ. Busto N, et al. Among authors: burke aj. RSC Med Chem. 2022 Jun 10;13(8):970-977. doi: 10.1039/d2md00044j. eCollection 2022 Aug 17. RSC Med Chem. 2022. PMID: 36092141 Free PMC article.

7

N-1,2,3-triazole-isatin derivatives for cholinesterase and β-amyloid aggregation inhibition: A comprehensive bioassay study.

Marques CS, López Ó, Bagetta D, Carreiro EP, Petralla S, Bartolini M, Hoffmann M, Alcaro S, Monti B, Bolognesi ML, Decker M, Fernández-Bolaños JG, Burke AJ. Marques CS, et al. Among authors: burke aj. Bioorg Chem. 2020 May;98:103753. doi: 10.1016/j.bioorg.2020.103753. Epub 2020 Mar 19. Bioorg Chem. 2020. PMID: 32200328

8

Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease.

Moutayakine A, Marques C, López Ó, Bagetta D, Leitzbach L, Hagenow S, Carreiro EP, Stark H, Alcaro S, Fernández-Bolaños JG, Burke AJ. Moutayakine A, et al. Among authors: burke aj. Bioorg Med Chem. 2022 Aug 15;68:116807. doi: 10.1016/j.bmc.2022.116807. Epub 2022 May 9. Bioorg Med Chem. 2022. PMID: 35653868

9

Metal-catalyzed coupling/carbonylative cyclizations for accessing dibenzodiazepinones: an expedient route to clozapine and other drugs.

Moutayakine A, Burke AJ. Moutayakine A, et al. Among authors: burke aj. Beilstein J Org Chem. 2024 Jan 31;20:193-204. doi: 10.3762/bjoc.20.19. eCollection 2024. Beilstein J Org Chem. 2024. PMID: 38318460 Free PMC article.

10

Asymmetric organocatalysis in drug discovery and development for active pharmaceutical ingredients.

Burke AJ. Burke AJ. Expert Opin Drug Discov. 2023 Jan;18(1):37-46. doi: 10.1080/17460441.2023.2160437. Epub 2022 Dec 26. Expert Opin Drug Discov. 2023. PMID: 36527181 Review.

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