Brigaud T - Search Results

1

Bimodal Use of Chiral α-Trifluoromethylalanine in Aib Foldamers: Study of the Position Impact Towards the Helical Screw-Sense Preference.

Picois N, Bodero L, Milbeo P, Brigaud T, Chaume G. Picois N, et al. Among authors: brigaud t. Chemistry. 2024 May 14;30(27):e202400540. doi: 10.1002/chem.202400540. Epub 2024 Mar 22. Chemistry. 2024. PMID: 38445775

2

Concise synthesis of enantiopure alpha-trifluoromethyl alanines, diamines, and amino alcohols via the Strecker-type reaction.

Huguenot F, Brigaud T. Huguenot F, et al. Among authors: brigaud t. J Org Chem. 2006 Sep 1;71(18):7075-8. doi: 10.1021/jo0607717. J Org Chem. 2006. PMID: 16930068

3

Convenient asymmetric synthesis of beta-trifluoromethyl-beta-amino acid, beta-amino ketones, and gamma-amino alcohols via Reformatsky and Mannich-type reactions from 2-trifluoromethyl-1,3-oxazolidines.

Huguenot F, Brigaud T. Huguenot F, et al. Among authors: brigaud t. J Org Chem. 2006 Mar 3;71(5):2159-62. doi: 10.1021/jo052323p. J Org Chem. 2006. PMID: 16497009

4

Umpolung reactivity of difluoroenol silyl ethers with amines and amino alcohols. application to the synthesis of enantiopure alpha-difluoromethyl amines and amino acids.

Huguenot F, Billac A, Brigaud T, Portella C. Huguenot F, et al. Among authors: brigaud t. J Org Chem. 2008 Apr 4;73(7):2564-9. doi: 10.1021/jo702328v. Epub 2008 Mar 11. J Org Chem. 2008. PMID: 18331052

5

Straightforward synthesis of (S)- and (R)-alpha-trifluoromethyl proline from chiral oxazolidines derived from ethyl trifluoropyruvate.

Chaume G, Van Severen MC, Marinkovic S, Brigaud T. Chaume G, et al. Among authors: brigaud t. Org Lett. 2006 Dec 21;8(26):6123-6. doi: 10.1021/ol062593+. Org Lett. 2006. PMID: 17165945

6

Iodocyclization of chiral CF3-allylmorpholinones: a versatile strategy for the synthesis of enantiopure alpha-Tfm-prolines and alpha-Tfm-dihydroxyprolines.

Caupène C, Chaume G, Ricard L, Brigaud T. Caupène C, et al. Among authors: brigaud t. Org Lett. 2009 Jan 1;11(1):209-12. doi: 10.1021/ol8024567. Org Lett. 2009. PMID: 19049401

7

Highly diastereoselective alpha-hydroxylation of Fox chiral auxiliary-based amide enolates with molecular oxygen.

Lubin H, Tessier A, Chaume G, Pytkowicz J, Brigaud T. Lubin H, et al. Among authors: brigaud t. Org Lett. 2010 Apr 2;12(7):1496-9. doi: 10.1021/ol100211s. Org Lett. 2010. PMID: 20218638

8

Synthesis of 2-trifluoromethyl-1,3-oxazolidines as hydrolytically stable pseudoprolines.

Chaume G, Barbeau O, Lesot P, Brigaud T. Chaume G, et al. Among authors: brigaud t. J Org Chem. 2010 Jun 18;75(12):4135-45. doi: 10.1021/jo100518t. J Org Chem. 2010. PMID: 20481551

9

Local control of the cis-trans isomerization and backbone dihedral angles in peptides using trifluoromethylated pseudoprolines.

Feytens D, Chaume G, Chassaing G, Lavielle S, Brigaud T, Byun BJ, Kang YK, Miclet E. Feytens D, et al. Among authors: brigaud t. J Phys Chem B. 2012 Apr 5;116(13):4069-79. doi: 10.1021/jp300284u. Epub 2012 Mar 22. J Phys Chem B. 2012. PMID: 22397724

10

Synthesis of an MIF-1 analogue containing enantiopure (S)-α-trifluoromethyl-proline and biological evaluation on nociception.

Jlalia I, Lensen N, Chaume G, Dzhambazova E, Astasidi L, Hadjiolova R, Bocheva A, Brigaud T. Jlalia I, et al. Among authors: brigaud t. Eur J Med Chem. 2013 Apr;62:122-9. doi: 10.1016/j.ejmech.2012.12.041. Epub 2013 Jan 3. Eur J Med Chem. 2013. PMID: 23353749

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