Reinoso RF - Search Results

1

WLB-87848, a Selective σ₁ Receptor Agonist, with an Unusually Positioned NH Group as Positive Ionizable Moiety and Showing Neuroprotective Activity.

Christmann U, Garriga L, Llorente AV, Díaz JL, Pascual R, Bordas M, Dordal A, Porras M, Yeste S, Reinoso RF, Vela JM, Almansa C. Christmann U, et al. Among authors: reinoso rf. J Med Chem. 2024 Jun 13;67(11):9150-9164. doi: 10.1021/acs.jmedchem.4c00288. Epub 2024 May 16. J Med Chem. 2024. PMID: 38753759

2

Discovery of WLB-89462, a New Drug-like and Highly Selective σ₂ Receptor Ligand with Neuroprotective Properties.

Christmann U, Díaz JL, Pascual R, Bordas M, Álvarez I, Monroy X, Porras M, Yeste S, Reinoso RF, Merlos M, Vela JM, Almansa C. Christmann U, et al. Among authors: reinoso rf. J Med Chem. 2023 Sep 14;66(17):12499-12519. doi: 10.1021/acs.jmedchem.3c01060. Epub 2023 Aug 22. J Med Chem. 2023. PMID: 37607512

3

Towards Multitargeted Ligands as Pain Therapeutics: Dual Ligands of the Ca_vα2δ-1 Subunit of Voltage-Gated Calcium Channel and the μ-Opioid Receptor.

Wegert A, Monnee M, de Graaf W, van Holst F, Bolcato G, Díaz JL, Dordal A, Portillo-Salido E, Reinoso RF, Yeste S, Torrens A, Almansa C. Wegert A, et al. Among authors: reinoso rf. ChemMedChem. 2024 May 17;19(10):e202300473. doi: 10.1002/cmdc.202300473. Epub 2024 Jan 17. ChemMedChem. 2024. PMID: 38230842

4

EST79232 and EST79376, Two Novel Sigma-1 Receptor Ligands, Exert Neuroprotection on Models of Motoneuron Degeneration.

Gaja-Capdevila N, Hernández N, Yeste S, Reinoso RF, Burgueño J, Montero A, Merlos M, Vela JM, Herrando-Grabulosa M, Navarro X. Gaja-Capdevila N, et al. Among authors: reinoso rf. Int J Mol Sci. 2022 Jun 16;23(12):6737. doi: 10.3390/ijms23126737. Int J Mol Sci. 2022. PMID: 35743175 Free PMC article.

5

Piperazinyl Bicyclic Derivatives as Selective Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels.

Fernández A, Díaz JL, García M, Rodríguez-Escrich S, Lorente A, Enrech R, Dordal A, Portillo-Salido E, Porras M, Fernández B, Reinoso RF, Vela JM, Almansa C. Fernández A, et al. Among authors: reinoso rf. ACS Med Chem Lett. 2021 Oct 5;12(11):1802-1809. doi: 10.1021/acsmedchemlett.1c00416. eCollection 2021 Nov 11. ACS Med Chem Lett. 2021. PMID: 34795870 Free PMC article.

6

Preliminary in vitro approach to evaluate the drug-drug interaction potential of EST73502, a dual µ-opioid receptor partial agonist and σ1 receptor antagonist.

Ayet E, Yeste S, Reinoso RF, Pretel MJ, Balada A, Serafini MT. Ayet E, et al. Among authors: reinoso rf. Xenobiotica. 2021 May;51(5):501-512. doi: 10.1080/00498254.2021.1877850. Epub 2021 Feb 23. Xenobiotica. 2021. PMID: 33622176

7

Bicyclic Diazepinones as Dual Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels and the Norepinephrine Transporter.

Díaz JL, Cuevas F, Pazos G, Álvarez-Bercedo P, Oliva AI, Sarmentero MÁ, Font D, Jiménez-Aquino A, Morón M, Port A, Pascual R, Dordal A, Portillo-Salido E, Reinoso RF, Vela JM, Almansa C. Díaz JL, et al. Among authors: reinoso rf. J Med Chem. 2021 Feb 25;64(4):2167-2185. doi: 10.1021/acs.jmedchem.0c01867. Epub 2021 Feb 16. J Med Chem. 2021. PMID: 33591743

8

Preliminary in vitro assessment of pharmacokinetic drug-drug interactions of EST64401 and EST64514, two sigma-1 receptor antagonists.

Reinoso RF, Yeste S, Ayet E, Pretel MJ, Balada A, Serafini MT. Reinoso RF, et al. Xenobiotica. 2021 Apr;51(4):373-386. doi: 10.1080/00498254.2020.1867332. Epub 2021 Jan 20. Xenobiotica. 2021. PMID: 33350877

9

Preliminary in Vitro Assessment of the Potential of EST64454, a Sigma-1 Receptor Antagonist, for Pharmacokinetic Drug-Drug Interactions.

Yeste S, Reinoso RF, Ayet E, Pretel MJ, Balada A, Serafini MT. Yeste S, et al. Among authors: reinoso rf. Biol Pharm Bull. 2020;43(1):68-76. doi: 10.1248/bpb.b19-00542. Biol Pharm Bull. 2020. PMID: 31902934 Free article.

10

Synthesis and pharmacological evaluation of fluorinated benzo[7]annulen-7-amines as GluN2B-selective NMDA receptor antagonists.

Thum S, Schepmann D, Reinoso RF, Alvarez I, Ametamey SM, Wünsch B. Thum S, et al. Among authors: reinoso rf. J Labelled Comp Radiopharm. 2019 Jun 30;62(8):354-379. doi: 10.1002/jlcr.3718. J Labelled Comp Radiopharm. 2019. PMID: 30850991

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