Loza MI - Search Results

1

N-Adamantyl-1-alkyl-4-oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as Fluorescent Probes to Detect Microglia Activation through the Imaging of Cannabinoid Receptor Subtype 2 (CB2R).

Intranuovo F, Majellaro M, Mastropasqua F, Delre P, Abatematteo FS, Mangiatordi GF, Stefanachi A, Brea J, Loza MI, Riganti C, Ligresti A, Kumar P, Esposito D, Cristino L, Nicois A, González L, Perrone MG, Colabufo NA, Sotelo E, Abate C, Contino M. Intranuovo F, et al. Among authors: loza mi. J Med Chem. 2024 Jul 11;67(13):11003-11023. doi: 10.1021/acs.jmedchem.4c00564. Epub 2024 Jun 27. J Med Chem. 2024. PMID: 38937147

2

Butyrophenone analogues in the carbazole series as potential atypical antipsychotics: synthesis and determination of affinities at D(2), 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.

Masaguer CF, Raviña E, Fontenla JA, Brea J, Tristán H, Loza MI. Masaguer CF, et al. Among authors: loza mi. Eur J Med Chem. 2000 Jan;35(1):83-95. doi: 10.1016/s0223-5234(00)00109-4. Eur J Med Chem. 2000. PMID: 10733606

3

New serotonin 5-HT(2A), 5-HT(2B), and 5-HT(2C) receptor antagonists: synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo and heterocycloalkanones.

Brea J, Rodrigo J, Carrieri A, Sanz F, Cadavid MI, Enguix MJ, Villazón M, Mengod G, Caro Y, Masaguer CF, Raviña E, Centeno NB, Carotti A, Loza MI. Brea J, et al. Among authors: loza mi. J Med Chem. 2002 Jan 3;45(1):54-71. doi: 10.1021/jm011014y. J Med Chem. 2002. PMID: 11754579

4

New arylpiperazine derivatives with high affinity for alpha1A, D2 and 5-HT2A receptors.

González-Gómez JC, Santana L, Uriarte E, Brea J, Villazón M, Loza MI, De Luca M, Rivas ME, Montenegro GY, Fontenla JA. González-Gómez JC, et al. Among authors: loza mi. Bioorg Med Chem Lett. 2003 Jan 20;13(2):175-8. doi: 10.1016/s0960-894x(02)00933-2. Bioorg Med Chem Lett. 2003. PMID: 12482418

5

Conformationally constrained butyrophenones as new pharmacological tools to study 5-HT 2A and 5-HT 2C receptor behaviours.

Brea J, Masaguer CF, Villazón M, Cadavid MI, Raviña E, Fontaine F, Dezi C, Pastor M, Sanz F, Loza MI. Brea J, et al. Among authors: loza mi. Eur J Med Chem. 2003 Apr;38(4):433-40. doi: 10.1016/s0223-5234(03)00054-0. Eur J Med Chem. 2003. PMID: 12750032

6

Synthesis and biological activity of new potential agonists for the human adenosine A2A receptor.

Bosch MP, Campos F, Niubó I, Rosell G, Díaz JL, Brea J, Loza MI, Guerrero A. Bosch MP, et al. Among authors: loza mi. J Med Chem. 2004 Jul 29;47(16):4041-53. doi: 10.1021/jm031143+. J Med Chem. 2004. PMID: 15267242

7

8-Substituted-9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B.

Carotti A, Stefanachi A, Raviña E, Sotelo E, Loza MI, Cadavid MI, Centeno NB, Nicolotti O. Carotti A, et al. Among authors: loza mi. Eur J Med Chem. 2004 Oct;39(10):879-87. doi: 10.1016/j.ejmech.2004.07.008. Eur J Med Chem. 2004. PMID: 15464622

8

Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor.

Carotti A, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Stefanachi A, Vidal B. Carotti A, et al. Among authors: loza mi. J Med Chem. 2006 Jan 12;49(1):282-99. doi: 10.1021/jm0506221. J Med Chem. 2006. PMID: 16392813

9

Multistructure 3D-QSAR studies on a series of conformationally constrained butyrophenones docked into a new homology model of the 5-HT2A receptor.

Dezi C, Brea J, Alvarado M, Raviña E, Masaguer CF, Loza MI, Sanz F, Pastor M. Dezi C, et al. Among authors: loza mi. J Med Chem. 2007 Jul 12;50(14):3242-55. doi: 10.1021/jm070277a. Epub 2007 Jun 19. J Med Chem. 2007. PMID: 17579386

10

1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor.

Stefanachi A, Brea JM, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Vidal B, Carotti A. Stefanachi A, et al. Among authors: loza mi. Bioorg Med Chem. 2008 Mar 15;16(6):2852-69. doi: 10.1016/j.bmc.2008.01.002. Epub 2008 Jan 10. Bioorg Med Chem. 2008. PMID: 18226909

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