Klein VG - Search Results

1

Picking the tyrosine-lock: chemical synthesis of the tyrosyl-DNA phosphodiesterase I inhibitor recifin A and analogues.

Smallwood TB, Krumpe LRH, Payne CD, Klein VG, O'Keefe BR, Clark RJ, Schroeder CI, Rosengren KJ. Smallwood TB, et al. Among authors: klein vg. Chem Sci. 2024 Jun 14;15(33):13227-13233. doi: 10.1039/d4sc01976h. eCollection 2024 Aug 22. Chem Sci. 2024. PMID: 39183914 Free PMC article.

2

Identifying the Cellular Target of Cordyheptapeptide A and Synthetic Derivatives.

Klein VG, Bray WM, Wang HY, Edmondson Q, Schwochert J, Ono S, Naylor MR, Turmon AC, Faris JH, Okada O, Taunton J, Lokey RS. Klein VG, et al. ACS Chem Biol. 2021 Aug 20;16(8):1354-1364. doi: 10.1021/acschembio.1c00094. Epub 2021 Jul 12. ACS Chem Biol. 2021. PMID: 34251165 Free PMC article.

3

Amide-to-Ester Substitution as a Strategy for Optimizing PROTAC Permeability and Cellular Activity.

Klein VG, Bond AG, Craigon C, Lokey RS, Ciulli A. Klein VG, et al. J Med Chem. 2021 Dec 23;64(24):18082-18101. doi: 10.1021/acs.jmedchem.1c01496. Epub 2021 Dec 9. J Med Chem. 2021. PMID: 34881891 Free PMC article.

4

Understanding and Improving the Membrane Permeability of VH032-Based PROTACs.

Klein VG, Townsend CE, Testa A, Zengerle M, Maniaci C, Hughes SJ, Chan KH, Ciulli A, Lokey RS. Klein VG, et al. ACS Med Chem Lett. 2020 Jul 30;11(9):1732-1738. doi: 10.1021/acsmedchemlett.0c00265. eCollection 2020 Sep 10. ACS Med Chem Lett. 2020. PMID: 32939229 Free PMC article.

5

Drug-Like Properties in Macrocycles above MW 1000: Backbone Rigidity versus Side-Chain Lipophilicity.

Furukawa A, Schwochert J, Pye CR, Asano D, Edmondson QD, Turmon AC, Klein VG, Ono S, Okada O, Lokey RS. Furukawa A, et al. Among authors: klein vg. Angew Chem Int Ed Engl. 2020 Nov 23;59(48):21571-21577. doi: 10.1002/anie.202004550. Epub 2020 Sep 17. Angew Chem Int Ed Engl. 2020. PMID: 32789999 Free PMC article.

6

Lipophilic Permeability Efficiency Reconciles the Opposing Roles of Lipophilicity in Membrane Permeability and Aqueous Solubility.

Naylor MR, Ly AM, Handford MJ, Ramos DP, Pye CR, Furukawa A, Klein VG, Noland RP, Edmondson Q, Turmon AC, Hewitt WM, Schwochert J, Townsend CE, Kelly CN, Blanco MJ, Lokey RS. Naylor MR, et al. Among authors: klein vg. J Med Chem. 2018 Dec 27;61(24):11169-11182. doi: 10.1021/acs.jmedchem.8b01259. Epub 2018 Dec 11. J Med Chem. 2018. PMID: 30395703

7

[ON THE SURGICAL TREATMENT OF CRYPTORCHISM].

POPOVIANTS RS, KLEIN VG, BORTNIKOV OG. POPOVIANTS RS, et al. Among authors: klein vg. Urol Mosc. 1964 May-Jun;29:13-6. Urol Mosc. 1964. PMID: 14225720 Russian. No abstract available.

8

[Treatment of varices of the spermatic cord].

KLEIN VG. KLEIN VG. Vestn Khir Im I I Grek. 1962 May;88:75-6. Vestn Khir Im I I Grek. 1962. PMID: 14456788 Russian. No abstract available.

9

[Acute paranephritis].

KLEIN VG. KLEIN VG. Urol Mosc. 1962 Mar-Apr;27:16-20. Urol Mosc. 1962. PMID: 14456787 Russian. No abstract available.

10

[Acute suppurative diseases of the retroperitoneal space of appendiceal etiology].

KLEIN VG, LEVINSKAIA BM. KLEIN VG, et al. Urol Mosc. 1961 Nov-Dec;26:26-7. Urol Mosc. 1961. PMID: 14456786 Russian. No abstract available.

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