Haemers A - Search Results

1

Dipeptide-derived diphenyl phosphonate esters: mechanism-based inhibitors of dipeptidyl peptidase IV.

Lambeir AM, Borloo M, De Meester I, Belyaev A, Augustyns K, Hendriks D, Scharpé S, Haemers A. Lambeir AM, et al. Among authors: haemers a. Biochim Biophys Acta. 1996 May 21;1290(1):76-82. doi: 10.1016/0304-4165(96)00012-8. Biochim Biophys Acta. 1996. PMID: 8645710

2

Development of potent and selective dipeptidyl peptidase II inhibitors.

Senten K, Van der Veken P, Bal G, De Meester I, Lambeir AM, Scharpé S, Bauvois B, Haemers A, Augustyns K. Senten K, et al. Among authors: haemers a. Bioorg Med Chem Lett. 2002 Oct 21;12(20):2825-8. doi: 10.1016/s0960-894x(02)00603-0. Bioorg Med Chem Lett. 2002. PMID: 12270155

3

Exploration of the active site of dipeptidyl peptidase IV from Porphyromonas gingivalis. Comparison with the human enzyme.

Lambeir AM, Rea D, Fülöp V, Kumagai Y, Augustyns K, de Meester I, Haemers A, Scharpé S. Lambeir AM, et al. Among authors: haemers a. Adv Exp Med Biol. 2003;524:29-35. doi: 10.1007/0-306-47920-6_3. Adv Exp Med Biol. 2003. PMID: 12675220 No abstract available.

4

Rapid parallel synthesis of dipeptide diphenyl phosphonate esters as inhibitors of dipeptidyl peptidases.

Senten K, Daniëls L, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: haemers a. J Comb Chem. 2003 May-Jun;5(3):336-44. doi: 10.1021/cc020096o. J Comb Chem. 2003. PMID: 12739951

5

Design, synthesis, and SAR of potent and selective dipeptide-derived inhibitors for dipeptidyl peptidases.

Senten K, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: haemers a. J Med Chem. 2003 Nov 6;46(23):5005-14. doi: 10.1021/jm0308803. J Med Chem. 2003. PMID: 14584950

6

Gamma-amino-substituted analogues of 1-[(S)-2,4-diaminobutanoyl]piperidine as highly potent and selective dipeptidyl peptidase II inhibitors.

Senten K, Van Der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: haemers a. J Med Chem. 2004 May 20;47(11):2906-16. doi: 10.1021/jm031122f. J Med Chem. 2004. PMID: 15139769

7

Prolyl peptidases related to dipeptidyl peptidase IV: potential of specific inhibitors in drug discovery.

Van der Veken P, Haemers A, Augustyns K. Van der Veken P, et al. Among authors: haemers a. Curr Top Med Chem. 2007;7(6):621-35. doi: 10.2174/156802607780091046. Curr Top Med Chem. 2007. PMID: 17352682 Review.

8

Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 1: identification of dipeptide derived leads.

Van der Veken P, De Meester I, Dubois V, Soroka A, Van Goethem S, Maes MB, Brandt I, Lambeir AM, Chen X, Haemers A, Scharpé S, Augustyns K. Van der Veken P, et al. Among authors: haemers a. Bioorg Med Chem Lett. 2008 Jul 15;18(14):4154-8. doi: 10.1016/j.bmcl.2008.05.080. Epub 2008 May 24. Bioorg Med Chem Lett. 2008. PMID: 18556199

9

The unique properties of dipeptidyl-peptidase IV (DPP IV / CD26) and the therapeutic potential of DPP IV inhibitors.

Augustyns K, Bal G, Thonus G, Belyaev A, Zhang XM, Bollaert W, Lambeir AM, Durinx C, Goossens F, Haemers A. Augustyns K, et al. Among authors: haemers a. Curr Med Chem. 1999 Apr;6(4):311-27. Curr Med Chem. 1999. PMID: 10101215 Review.

10

Study of the enzymatic degradation of vasostatin I and II and their precursor chromogranin A by dipeptidyl peptidase IV using high-performance liquid chromatography/electrospray mass spectrometry.

Zhang XY, De Meester I, Lambeir AM, Dillen L, Van Dongen W, Esmans EL, Haemers A, Scharpé S, Claeys M. Zhang XY, et al. Among authors: haemers a. J Mass Spectrom. 1999 Apr;34(4):255-63. doi: 10.1002/(SICI)1096-9888(199904)34:4<255::AID-JMS752>3.0.CO;2-7. J Mass Spectrom. 1999. PMID: 10226356

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