Bousquet P - Search Results

1

Imidazoline receptors: qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity.

Pigini M, Bousquet P, Carotti A, Dontenwill M, Giannella M, Moriconi R, Piergentili A, Quaglia W, Tayebati SK, Brasili L. Pigini M, et al. Among authors: bousquet p. Bioorg Med Chem. 1997 May;5(5):833-41. doi: 10.1016/s0968-0896(97)00009-6. Bioorg Med Chem. 1997. PMID: 9208095

2

Alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole.

Gentili F, Bousquet P, Brasili L, Caretto M, Carrieri A, Dontenwill M, Giannella M, Marucci G, Perfumi M, Piergentili A, Quaglia W, Rascente C, Pigini M. Gentili F, et al. Among authors: bousquet p. J Med Chem. 2002 Jan 3;45(1):32-40. doi: 10.1021/jm0110082. J Med Chem. 2002. PMID: 11754577

3

Imidazoline binding sites (IBS) profile modulation: key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues.

Gentili F, Bousquet P, Brasili L, Dontenwill M, Feldman J, Ghelfi F, Giannella M, Piergentili A, Quaglia W, Pigini M. Gentili F, et al. Among authors: bousquet p. J Med Chem. 2003 May 22;46(11):2169-76. doi: 10.1021/jm021113r. J Med Chem. 2003. PMID: 12747788

4

2-D and 3-D modeling of imidazoline receptor ligands: insights into pharmacophore.

Carrieri A, Brasili L, Leonetti F, Pigini M, Giannella M, Bousquet P, Carotti A. Carrieri A, et al. Among authors: bousquet p. Bioorg Med Chem. 1997 May;5(5):843-56. doi: 10.1016/s0968-0896(97)00023-0. Bioorg Med Chem. 1997. PMID: 9208096

5

Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models.

Pigini M, Bousquet P, Brasili L, Carrieri A, Cavagna R, Dontenwill M, Gentili F, Giannella M, Leonetti F, Piergentili A, Quaglia W, Carotti A. Pigini M, et al. Among authors: bousquet p. Bioorg Med Chem. 1998 Dec;6(12):2245-60. doi: 10.1016/s0968-0896(98)80005-9. Bioorg Med Chem. 1998. PMID: 9925287

6

Binding of tracizolines to the imidazoline receptor. Role of lipophilicity in quantitative structure-activity relationship models.

Pigini M, Bousquet P, Brasili L, Carrieri A, Dontenwill M, Gentili F, Giannella M, Leonetti F, Piergentili A, Quaglia W, Carotti A. Pigini M, et al. Among authors: bousquet p. Ann N Y Acad Sci. 1999 Jun 21;881:118-22. doi: 10.1111/j.1749-6632.1999.tb09351.x. Ann N Y Acad Sci. 1999. PMID: 10415907 No abstract available.

7

2-(2-Phenylcyclopropyl)imidazolines: reversed enantioselective interaction at I(1) and I(2) imidazoline receptors.

Quaglia W, Bousquet P, Pigini M, Carotti A, Carrieri A, Dontenwill M, Gentili F, Giannella M, Maranca F, Piergentili A, Brasili L. Quaglia W, et al. Among authors: bousquet p. J Med Chem. 1999 Jul 29;42(15):2737-40. doi: 10.1021/jm991049m. J Med Chem. 1999. PMID: 10425083 No abstract available.

8

Methylation of imidazoline related compounds leads to loss of α₂-adrenoceptor affinity. Synthesis and biological evaluation of selective I₁ imidazoline receptor ligands.

Schann S, Greney H, Gasparik V, Dontenwill M, Rascente C, Lacroix G, Monassier L, Bruban V, Feldman J, Ehrhardt JD, Bousquet P. Schann S, et al. Among authors: bousquet p. Bioorg Med Chem. 2012 Aug 1;20(15):4710-5. doi: 10.1016/j.bmc.2012.06.008. Epub 2012 Jun 9. Bioorg Med Chem. 2012. PMID: 22750139

9

Structure-affinity relationship of cirazoline derivatives for idazoxan imidazoline-specific sites in the human cerebral cortex and the rabbit kidney.

Brasili L, Pigini M, Ehrhardt JD, Molines A, Greney H, Bousquet P, Dontenwill M. Brasili L, et al. Among authors: bousquet p. Ann N Y Acad Sci. 1995 Jul 12;763:149-52. doi: 10.1111/j.1749-6632.1995.tb32399.x. Ann N Y Acad Sci. 1995. PMID: 7677323 No abstract available.

10

I1-imidazoline receptors: an update.

Bousquet P, Dontenwill M, Greney H, Feldman J. Bousquet P, et al. J Hypertens Suppl. 1998 Aug;16(3):S1-5. J Hypertens Suppl. 1998. PMID: 9747903 Review.

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