Glucose hypometabolism prompts RAN translation and exacerbates C9orf72-related ALS/FTD phenotypes

EMBO Rep. 2024 May;25(5):2479-2510. doi: 10.1038/s44319-024-00140-7. Epub 2024 Apr 29.

Abstract

The most prevalent genetic cause of both amyotrophic lateral sclerosis and frontotemporal dementia is a (GGGGCC)n nucleotide repeat expansion (NRE) occurring in the first intron of the C9orf72 gene (C9). Brain glucose hypometabolism is consistently observed in C9-NRE carriers, even at pre-symptomatic stages, but its role in disease pathogenesis is unknown. Here, we show alterations in glucose metabolic pathways and ATP levels in the brains of asymptomatic C9-BAC mice. We find that, through activation of the GCN2 kinase, glucose hypometabolism drives the production of dipeptide repeat proteins (DPRs), impairs the survival of C9 patient-derived neurons, and triggers motor dysfunction in C9-BAC mice. We also show that one of the arginine-rich DPRs (PR) could directly contribute to glucose metabolism and metabolic stress by inhibiting glucose uptake in neurons. Our findings provide a potential mechanistic link between energy imbalances and C9-ALS/FTD pathogenesis and suggest a feedforward loop model with potential opportunities for therapeutic intervention.

Keywords: ALS; C9orf72; FTD; Glucose Hypometabolism; RAN Translation.

MeSH terms

  • Adenosine Triphosphate / metabolism
  • Amyotrophic Lateral Sclerosis* / genetics
  • Amyotrophic Lateral Sclerosis* / metabolism
  • Amyotrophic Lateral Sclerosis* / pathology
  • Animals
  • Brain / metabolism
  • Brain / pathology
  • C9orf72 Protein* / genetics
  • C9orf72 Protein* / metabolism
  • DNA Repeat Expansion / genetics
  • Disease Models, Animal
  • Frontotemporal Dementia* / genetics
  • Frontotemporal Dementia* / metabolism
  • Frontotemporal Dementia* / pathology
  • Glucose* / metabolism
  • Mice
  • Mice, Transgenic
  • Neurons / metabolism
  • Phenotype*
  • Protein Biosynthesis
  • ran GTP-Binding Protein* / metabolism

Substances

  • Adenosine Triphosphate
  • C9orf72 Protein
  • Glucose
  • Ran protein, mouse
  • ran GTP-Binding Protein