The spectral and thermodynamic properties of staphylococcal enterotoxin A, E, and variants suggest that structural modifications are important to control their function

J Biol Chem. 2000 Jan 21;275(3):1665-72. doi: 10.1074/jbc.275.3.1665.

Abstract

The superantigens staphylococcal enterotoxin A and E (SEA and SEE) can activate a large number of T-cells. SEA and SEE have approximately 80% sequence identity but show some differences in their biological function. Here, the two superantigens and analogues were characterized biophysically. SEE was shown to have a substantially higher thermal stability than SEA. Both SEA and SEE were thermally stabilized by 0.1 mM Zn(2+) compared with Zn(2+)-reduced conditions achieved using 1 mM EDTA or specific replacements that affect Zn(2+) coordination. The higher stability of SEE was only partly caused by the T-cell receptor (TCR) binding regions, whereas regions in the vicinity of the major histocompatibility complex class II binding sites affected the stability to a greater extent. SEE exhibited a biphasic denaturation between pH 5.0-6.5, influenced by residues in the TCR binding regions. Interestingly, enzyme-linked immunosorbent assay, isoelectric focusing, and circular dichroism analysis indicated that conformational changes had occurred in the SEA/E chimerical constructs relative to SEA and SEE. Thus, it is proposed that the Zn(2+) binding site is very important for the stability and potency of SEA and SEE, whereas residues in the TCR binding site have a substantial influence on the molecular conformation to control specificity and function.

Publication types

  • Comparative Study

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Cells, Cultured
  • Circular Dichroism
  • Dose-Response Relationship, Drug
  • Enterotoxins / chemistry*
  • Guanidine / pharmacology
  • Histocompatibility Antigens Class II / metabolism
  • Hydrogen-Ion Concentration
  • Mice
  • Mice, Inbred C57BL
  • Molecular Sequence Data
  • Protein Binding
  • Protein Denaturation
  • Protein Structure, Tertiary
  • Recombinant Fusion Proteins / chemistry
  • Sequence Homology, Amino Acid
  • Spleen / metabolism
  • Structure-Activity Relationship
  • Superantigens / metabolism
  • T-Lymphocytes / metabolism
  • Temperature
  • Thermodynamics
  • Zinc / metabolism

Substances

  • Enterotoxins
  • Histocompatibility Antigens Class II
  • Recombinant Fusion Proteins
  • Superantigens
  • enterotoxin E, Staphylococcal
  • enterotoxin A, Staphylococcal
  • Zinc
  • Guanidine