The roles of E6-AP and MDM2 in p53 regulation in human papillomavirus-positive cervical cancer cells

Antisense Nucleic Acid Drug Dev. 2000 Feb;10(1):17-27. doi: 10.1089/oli.1.2000.10.17.

Abstract

The p53 tumor suppressor is regulated by the MDM2 oncoprotein through a negative feedback mechanism. MDM2 promotes the ubiquitination and proteasome-dependent degradation of p53, possibly by acting as a ubiquitin ligase. In cervical cancer cells containing high-risk human papillomaviruses (HPV), p53 is also targeted for degradation by the HPV E6 oncoprotein in combination with the cellular E6-AP ubiquitin ligase. In this report, we describe the identification of efficient antisense oligonucleotides against human E6-AP. The roles of MDM2 and E6-AP in p53 regulation were investigated using a novel E6-AP antisense oligonucleotide and a previously characterized MDM2 antisense oligonucleotide. In HPV16-positive and HPV-18 positive cervical cancer cells, inhibition of E6-AP, but not MDM2, expression results in significant induction of p53. In HPV-negative tumor cells, p53 is activated by inhibition of MDM2 but not E6-AP. Furthermore, treatment with both E6-AP and MDM2 antisense oligonucleotides in HPV-positive cells does not lead to further induction of p53 over inhibition of E6-AP alone. Therefore, E6-AP-mediated degradation is dominant over MDM2 in cervical cancer cells but does not have a significant role in HPV-negative cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Survival / drug effects
  • Doxorubicin / pharmacology
  • Female
  • Fluorescent Antibody Technique
  • Gene Expression Regulation, Neoplastic / drug effects
  • Humans
  • Ligases / antagonists & inhibitors
  • Ligases / genetics
  • Ligases / metabolism*
  • Nuclear Proteins*
  • Oligonucleotides, Antisense / pharmacology
  • Papillomaviridae / genetics*
  • Phosphatidylethanolamines / metabolism
  • Proto-Oncogene Proteins / antagonists & inhibitors
  • Proto-Oncogene Proteins / genetics
  • Proto-Oncogene Proteins / metabolism*
  • Proto-Oncogene Proteins c-mdm2
  • RNA, Messenger / metabolism
  • Tumor Cells, Cultured
  • Tumor Suppressor Protein p53 / metabolism*
  • Ubiquitin-Protein Ligases
  • Uterine Cervical Neoplasms / virology

Substances

  • Nuclear Proteins
  • Oligonucleotides, Antisense
  • Phosphatidylethanolamines
  • Proto-Oncogene Proteins
  • RNA, Messenger
  • Tumor Suppressor Protein p53
  • 1,2-dielaidoylphosphatidylethanolamine
  • Doxorubicin
  • MDM2 protein, human
  • Proto-Oncogene Proteins c-mdm2
  • Ubiquitin-Protein Ligases
  • Ligases