Ligand-presenting assembly: a method for C- and N-terminal antigen presentation

J Pept Res. 2000 Aug;56(2):105-13. doi: 10.1034/j.1399-3011.2000.00758.x.

Abstract

Achiral dicarboxylic acids were coupled with 2 eq. of the free alpha-amino groups of two fully side-chain protected peptide chains while these were still attached to a synthesis resin. Cleavage from the resin with simultaneous side-chain deprotection afforded two assembled peptide chains with free C-terminals. Suitable functionalization of the achiral dicarboxylic acid alternatively permitted continued peptide synthesis in a C to N orientation leading to a final peptide assembly which, after cleavage from the resin, may have multiple N to C and C to N presentation of one or more epitopes.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antigens, Bacterial / biosynthesis
  • Antigens, Bacterial / chemistry
  • Antigens, Bacterial / immunology*
  • Borrelia / immunology
  • Carbon / chemistry
  • Chromatography, High Pressure Liquid
  • Enzyme-Linked Immunosorbent Assay
  • Epitopes, B-Lymphocyte / chemistry*
  • Ligands
  • Mice
  • Molecular Sequence Data
  • Nitrogen / chemistry

Substances

  • Antigens, Bacterial
  • Epitopes, B-Lymphocyte
  • Ligands
  • Carbon
  • Nitrogen