Runx2 is a common target of transforming growth factor beta1 and bone morphogenetic protein 2, and cooperation between Runx2 and Smad5 induces osteoblast-specific gene expression in the pluripotent mesenchymal precursor cell line C2C12

Mol Cell Biol. 2000 Dec;20(23):8783-92. doi: 10.1128/MCB.20.23.8783-8792.2000.

Abstract

When C2C12 pluripotent mesenchymal precursor cells are treated with transforming growth factor beta1 (TGF-beta1), terminal differentiation into myotubes is blocked. Treatment with bone morphogenetic protein 2 (BMP-2) not only blocks myogenic differentiation of C2C12 cells but also induces osteoblast differentiation. The molecular mechanisms governing the ability of TGF-beta1 and BMP-2 to both induce ligand-specific responses and inhibit myogenic differentiation are not known. We identified Runx2/PEBP2alphaA/Cbfa1, a global regulator of osteogenesis, as a major TGF-beta1-responsive element binding protein induced by TGF-beta1 and BMP-2 in C2C12 cells. Consistent with the observation that Runx2 can be induced by either TGF-beta1 or BMP-2, the exogenous expression of Runx2 mediated some of the effects of TGF-beta1 and BMP-2 but not osteoblast-specific gene expression. Runx2 mimicked common effects of TGF-beta1 and BMP-2 by inducing expression of matrix gene products (for example, collagen and fibronectin), suppressing MyoD expression, and inhibiting myotube formation of C2C12 cells. For osteoblast differentiation, an additional effector, BMP-specific Smad protein, was required. Our results indicate that Runx2 is a major target gene shared by TGF-beta and BMP signaling pathways and that the coordinated action of Runx2 and BMP-activated Smads leads to the induction of osteoblast-specific gene expression in C2C12 cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Bone Morphogenetic Protein 2
  • Bone Morphogenetic Proteins / pharmacology*
  • Cell Differentiation
  • Cell Line
  • Core Binding Factor Alpha 1 Subunit
  • DNA-Binding Proteins / metabolism*
  • Gene Expression Regulation, Developmental
  • Mesoderm / cytology*
  • Mesoderm / drug effects
  • Mice
  • Models, Biological
  • Neoplasm Proteins*
  • Osteoblasts / cytology*
  • Osteogenesis / physiology
  • Phosphoproteins / metabolism*
  • Protein Binding
  • Response Elements
  • Smad5 Protein
  • Stem Cells / cytology
  • Stem Cells / drug effects
  • Trans-Activators / metabolism*
  • Transcription Factors / metabolism*
  • Transforming Growth Factor beta / pharmacology*
  • Transforming Growth Factor beta1

Substances

  • Bmp2 protein, mouse
  • Bone Morphogenetic Protein 2
  • Bone Morphogenetic Proteins
  • Core Binding Factor Alpha 1 Subunit
  • DNA-Binding Proteins
  • Neoplasm Proteins
  • Phosphoproteins
  • Smad5 Protein
  • Smad5 protein, mouse
  • Tgfb1 protein, mouse
  • Trans-Activators
  • Transcription Factors
  • Transforming Growth Factor beta
  • Transforming Growth Factor beta1