The enzymatic activity of ADAM8 and ADAM9 is not regulated by TIMPs

FEBS Lett. 2002 Jul 31;524(1-3):154-8. doi: 10.1016/s0014-5793(02)03047-8.

Abstract

The ADAM family of proteases are type I transmembrane proteins with both metalloproteinase and disintegrin containing extracellular domains. ADAMs are implicated in the proteolytic processing of membrane-bound precursors and involved in modulating cell-cell and cell-matrix interactions. ADAM8 (MS2, CD156) has been identified in myeloid and B cells. In this report we demonstrate that soluble ADAM8 is an active metalloprotease in vitro and is able to hydrolyse myelin basic protein and a variety of peptide substrates based on the cleavage sites of membrane-bound cytokines, growth factors and receptors which are known to be processed by metalloproteinases. Interestingly, although ADAM8 was inhibited by a number of peptide analogue hydroxamate inhibitors, it was not inhibited by the tissue inhibitors of metalloproteinases (TIMPs). We also demonstrate that the activity of recombinant soluble ADAM9 (meltrin-gamma, MDC9) lacks inhibition by the TIMPs, but can be inhibited by hydroxamate inhibitors. The lack of TIMP inhibition of ADAM8 and 9 contrasts with other membrane-associated metalloproteinases characterised to date in this respect (ADAM10, 12, 17, and the membrane-type metalloproteinases) which have been implicated in protein processing at the cell surface.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • ADAM Proteins
  • Amino Acid Sequence
  • Antigens, CD*
  • Antigens, Surface / genetics
  • Antigens, Surface / isolation & purification
  • Antigens, Surface / metabolism*
  • Catalysis
  • Chromatography, Affinity
  • Disintegrins / metabolism*
  • Electrophoresis, Polyacrylamide Gel
  • Membrane Proteins*
  • Metalloendopeptidases / antagonists & inhibitors
  • Metalloendopeptidases / genetics
  • Metalloendopeptidases / isolation & purification
  • Metalloendopeptidases / metabolism*
  • Molecular Sequence Data
  • Recombinant Proteins / isolation & purification
  • Recombinant Proteins / metabolism
  • Tissue Inhibitor of Metalloproteinases / metabolism*

Substances

  • Antigens, CD
  • Antigens, Surface
  • Disintegrins
  • Membrane Proteins
  • Recombinant Proteins
  • Tissue Inhibitor of Metalloproteinases
  • ADAM Proteins
  • ADAM9 protein, human
  • Metalloendopeptidases