Identification of functional hypoxia response elements in the promoter region of the DEC1 and DEC2 genes

J Biol Chem. 2002 Dec 6;277(49):47014-21. doi: 10.1074/jbc.M204938200. Epub 2002 Sep 26.

Abstract

Adaptation to hypoxia is a crucial process both physiologically (i.e. in chondrocytes) and pathologically (i.e. in tumor cells). Previous studies have shown that DEC1, a basic helix-loop-helix transcription factor, is induced by hypoxia in glioma cells (Ivanova, A. V., Ivanov, S. V., Danilkovitch-Miagkova, A., and Lerman, M. I. (2001) J. Biol. Chem. 276, 15306-15315). In the present study, we found that hypoxia or CoCl(2) enhanced the mRNA expression of DEC2, as well as DEC1, within 24 h in chondrogenic ATDC5, 293T, and HeLa cells. In luciferase assays, the regions between -524 and -401 in the DEC1 promoter, and between -863 and -258 in the DEC2 promoter, were responsible for the hypoxia- or hypoxia-inducible factor-1alpha (HIF-1alpha)-induced transcription. In these regions, we identified functional hypoxia response elements (HREs) that bound to HIF-1alpha and HIF-1beta. In addition to an HIF-1 binding site consensus sequence, the DEC1 HRE had cAMP response element-like and CACAG sequences, which were also involved in the transcription activation in response to HIF-1alpha. Although the DEC2 HRE did not have a cAMP response element-like or CACAG sequence, it showed a higher affinity for HIF-1 than did the DEC1 HRE. Because DEC1 and DEC2 are directly inducible by HIF-1, these transcription factors may be crucial for the adaptation to hypoxia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aryl Hydrocarbon Receptor Nuclear Translocator
  • Base Sequence
  • Basic Helix-Loop-Helix Transcription Factors
  • Binding Sites
  • Cell Line
  • Cell Nucleus / metabolism
  • Chondrocytes / metabolism
  • Cobalt / metabolism
  • Collagen / metabolism
  • Cyclic AMP / metabolism
  • DNA-Binding Proteins*
  • HeLa Cells
  • Homeodomain Proteins / genetics*
  • Humans
  • Hypoxia
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • Luciferases / metabolism
  • Molecular Sequence Data
  • Oxidation-Reduction*
  • Plasmids / metabolism
  • Promoter Regions, Genetic*
  • RNA, Messenger / metabolism
  • Receptors, Aryl Hydrocarbon*
  • Response Elements*
  • Reverse Transcriptase Polymerase Chain Reaction
  • Time Factors
  • Transcription Factors / genetics*
  • Transcription Factors / metabolism
  • Transcription, Genetic
  • Transfection

Substances

  • ARNT protein, human
  • BHLHE40 protein, human
  • BHLHE41 protein, human
  • Basic Helix-Loop-Helix Transcription Factors
  • DNA-Binding Proteins
  • HIF1A protein, human
  • Homeodomain Proteins
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • RNA, Messenger
  • Receptors, Aryl Hydrocarbon
  • Transcription Factors
  • Aryl Hydrocarbon Receptor Nuclear Translocator
  • Cobalt
  • Collagen
  • Cyclic AMP
  • Luciferases
  • cobaltous chloride