Effect of thalidomide in patients with chronic heart failure

Am Heart J. 2002 Nov;144(5):847-50. doi: 10.1067/mhj.2002.125628.

Abstract

Background: Congestive heart failure (CHF) is characterized by enhanced immune activation, which possibly plays a pathogenic role in this disorder. We therefore examined whether immunomodulation with thalidomide could improve cardiac performance in patients with CHF.

Methods: Nine patients with chronic symptomatic CHF and left ventricular ejection fraction (LVEF) <40%, who were receiving "optimal" conventional cardiovascular treatment, were given 200 mg thalidomide daily in an open design for a period of 6 weeks. Tumor necrosis factor (TNF)-alpha and LVEF were measured at baseline and on completion of the study.

Results: Two patients withdrew because of side effects. Sedation was common and required dose reduction in 6 of 7 patients completing the study. Plasma levels of TNF-alpha were elevated at baseline compared with levels in healthy control patients, but decreased significantly from 33.9 +/- 10.1 pg/mL to 19.3 +/- 6.1 pg/mL during therapy (P <.05). LVEF increased in all patients from 26% +/- 9% to 34% +/- 10% at the end of the observation period (P <.05).

Conclusions: In this pilot study, therapy with thalidomide in patients with CHF resulted in decreased TNF-alpha levels and increased cardiac performance. Although few patients were included, our results suggest that thalidomide should be further investigated as an immunomodulating agent in CHF.

MeSH terms

  • Aged
  • Biomarkers / blood
  • Female
  • Heart Failure / blood
  • Heart Failure / drug therapy*
  • Heart Failure / immunology
  • Humans
  • Hypnotics and Sedatives / adverse effects
  • Hypnotics and Sedatives / therapeutic use
  • Immunosuppressive Agents / adverse effects
  • Immunosuppressive Agents / therapeutic use*
  • Male
  • Pilot Projects
  • Stroke Volume / drug effects
  • Thalidomide / adverse effects
  • Thalidomide / therapeutic use*
  • Tumor Necrosis Factor-alpha / drug effects
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Biomarkers
  • Hypnotics and Sedatives
  • Immunosuppressive Agents
  • Tumor Necrosis Factor-alpha
  • Thalidomide