Scabrolides A-D, four new norditerpenoids isolated from the soft coral Sinularia scabra

J Nat Prod. 2002 Dec;65(12):1904-8. doi: 10.1021/np020280r.

Abstract

Four new norditerpenoids, scabrolides A-D (1-4), along with four known ones, 5-8, have been isolated from the dichloromethane extract of the Taiwanese soft coral Sinularia scabra. The structures of 1-4 were elucidated on the basis of extensive spectroscopic analyses, while the relative configurations were determined by the NOESY experiments. The epimeric metabolites 6 and 7 have been shown to exhibit strong cytotoxic activity against KB and Hepa59T/VGH cancer cell lines.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anthozoa / chemistry*
  • Diterpenes / chemistry
  • Diterpenes / isolation & purification*
  • Diterpenes / pharmacology
  • Drug Screening Assays, Antitumor
  • Gas Chromatography-Mass Spectrometry
  • Humans
  • KB Cells / drug effects
  • Methylene Chloride
  • Molecular Conformation
  • Molecular Structure
  • Nuclear Magnetic Resonance, Biomolecular
  • Stereoisomerism
  • Taiwan
  • Tumor Cells, Cultured / drug effects

Substances

  • Diterpenes
  • Methylene Chloride