p53 Activation in adipocytes of obese mice

J Biol Chem. 2003 Jul 11;278(28):25395-400. doi: 10.1074/jbc.M302364200. Epub 2003 May 6.

Abstract

The tumor suppressor p53 is a transcription factor that activates or represses its target genes after various genotoxic stresses. We have previously shown that sterol regulatory element-binding protein-1 (SREBP-1), a key transcriptional regulator of triglyceride synthesis, and the lipogenic enzymes under its control are markedly suppressed in adipocytes from genetically obese ob/ob mice. Here we demonstrate that p53 and its target genes are highly induced in adipocytes of ob/ob mice in a fed state, leading to the negative regulation of SREBP-1 and thereby lipogenic genes. In fact, disruption of p53 in ob/ob mice completely suppressed the p53-regulated genes to wild-type levels and partially restored expression of lipogenic enzymes. Consistently, reporter gene analysis showed that p53 overexpression suppressed the promoter activity of the SREBP-1c gene and its downstream genes. Thus, the activation of p53 might constitute a negative feedback loop against excess fat accumulation in adipocytes. In conclusion, we discovered a novel role of p53 in the pathophysiology of obesity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adipose Tissue / metabolism
  • Animals
  • Blotting, Northern
  • Blotting, Western
  • CCAAT-Enhancer-Binding Proteins / metabolism*
  • Cell Nucleus / metabolism
  • Crosses, Genetic
  • DNA-Binding Proteins / metabolism*
  • Down-Regulation
  • Gene Expression Regulation*
  • Genotype
  • Immunoblotting
  • Luciferases / metabolism
  • Mice
  • Mice, Inbred C57BL
  • Mice, Obese
  • Obesity / metabolism
  • Plasmids / metabolism
  • Promoter Regions, Genetic
  • RNA, Messenger / metabolism
  • Sterol Regulatory Element Binding Protein 1
  • Transcription Factors*
  • Transcription, Genetic
  • Transfection
  • Tumor Suppressor Protein p53 / metabolism*
  • Up-Regulation

Substances

  • CCAAT-Enhancer-Binding Proteins
  • DNA-Binding Proteins
  • RNA, Messenger
  • Srebf1 protein, mouse
  • Sterol Regulatory Element Binding Protein 1
  • Transcription Factors
  • Tumor Suppressor Protein p53
  • Luciferases