Retinoic acid stimulates chondrocyte differentiation and enhances bone morphogenetic protein effects through induction of Smad1 and Smad5

Endocrinology. 2003 Jun;144(6):2514-23. doi: 10.1210/en.2002-220969.

Abstract

Whereas bone morphogenetic protein (BMP)-signaling events induce maturational characteristics in vitro, recent evidence suggests that the effects of other regulators might be mediated through BMP-signaling events. The present study examines the mechanism through which retinoic acid (RA) stimulates differentiation in chicken embryonic caudal sternal chondrocyte cultures. Both RA and BMP-2 induced expression of the chondrocyte maturational marker, colX, in chondrocyte cultures by 8 d. Though the RA effect was small, it synergistically enhanced the effect of BMP-2 on colX and phosphatase activity. Inhibition of either RA or BMP signaling, with selective inhibitors, interfered with the inductive effects of these agents but also inhibited the complementary pathway, demonstrating a codependence of RA and BMP signaling during chondrocyte maturation. BMP-2 did not enhance the effects of RA on an RA-responsive reporter construct, but RA enhanced basal activity and synergistically enhanced BMP-2 stimulation of the BMP-responsive chicken type X collagen reporter. A similar synergistic interaction between RA and BMP-2 was observed on colX expression. RA did not increase the expression of the type IA BMP receptor but did markedly up-regulate the expression of Smad1 and Smad5 proteins, important participants in the BMP pathway. Inhibition of RA signaling, with the selective inhibitor AGN 193109, blocked RA-mediated induction of the Smad proteins and chondrocyte differentiation. These findings demonstrate that RA induces the expression of BMP-signaling molecules and enhances BMP effects in chondrocytes.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alkaline Phosphatase / metabolism
  • Animals
  • Antineoplastic Agents / pharmacology*
  • Bone Morphogenetic Protein 2
  • Bone Morphogenetic Proteins / pharmacology*
  • Cell Differentiation / drug effects
  • Chick Embryo
  • Chickens
  • Chondrocytes / cytology*
  • Chondrocytes / physiology
  • Collagen Type X / genetics
  • DNA-Binding Proteins / genetics*
  • Drug Synergism
  • Phosphoproteins / genetics
  • Signal Transduction / drug effects
  • Smad Proteins
  • Smad5 Protein
  • Sternum / cytology
  • Trans-Activators / genetics*
  • Transforming Growth Factor beta*
  • Tretinoin / pharmacology*

Substances

  • Antineoplastic Agents
  • Bone Morphogenetic Protein 2
  • Bone Morphogenetic Proteins
  • Collagen Type X
  • DNA-Binding Proteins
  • Phosphoproteins
  • Smad Proteins
  • Smad5 Protein
  • Trans-Activators
  • Transforming Growth Factor beta
  • Tretinoin
  • Alkaline Phosphatase